SCHEMBL12411511

SCHEMBL12411511

[C-]#[N+]c1cc2c(Oc3ccc(NC(=O)Nc4nccs4)cc3)ccnc2cc1OCCCN1CCOCC1

nearest known ligand 0.54

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MET P08581 17/20 0.54
KDR P35968 1/20 0.54
RET P07949 1/20 0.53
EGFR P00533 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12411487 0.90 MET (0.60) METKDRRETEGFR
SCHEMBL12411362 0.90 MET (0.67) METKDRRETEGFR
SCHEMBL12411326 0.90 MET (0.63) METKDREGFR
SCHEMBL1896688 0.88 MET (0.54) METKDRRETEGFR
SCHEMBL12411414 0.88 MET (0.60) METKDREGFR
SCHEMBL12411454 0.86 FGFR2 (0.60) METKDREGFR
SCHEMBL12411484 0.84 FLT3 (0.55) METKDRRETEGFR
SCHEMBL12411331 0.84 PDGFRA (0.54) METKDR
SCHEMBL12411782 0.84 MET (0.60) METKDRRETEGFR
SCHEMBL12412260 0.83 KDR (0.55) METKDRRETEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7973160-B2 Nitrogen-containing aromatic derivatives EISAI R&D MANAGEMENT CO., LTD. (JP) 2011-07-05 US disclosed
US-20100197911-A1 Nitrogen-Containing Aromatic Derivatives EISAI R&D MANAGEMENT CO., LTD. (JP) 2010-08-05 US disclosed
US-7612092-B2 Urea derivatives containing aromatic or heteroaromatic rings; 4-(3-chloro-4-(cyclopropylaminocarbonyl)aminophenoxy)-7-methoxy-6-quinolinecarboxamide; prophylactic or therapeutic agent for a disease for which angiogenesis inhibition is effective EISAI R & D MANAGEMENT CO., LTD. (JP) 2009-11-03 US disclosed
US-7253286-B2 Urea derivatives containing aromatic or heteroaromatic rings, useful as prophylactic or therapeutic agent for a disease for which angiogenesis inhibition is effective EISAI CO., LTD (JP) 2007-08-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100197911-A1 Nitrogen-Containing Aromatic Derivatives GNG2, GCG, FRG1 MET 1810/4885KDR 2687/4885RET 1840/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.