SCHEMBL1241183

SCHEMBL1241183

CC(c1ccc(I)cc1)[C@H](NC(=O)OC(C)(C)C)C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CTSK P43235 5/20 0.41
CTSS P25774 3/20 0.41
TRPA1 O75762 2/20 0.41
APP P05067 2/20 0.39
PPARA Q07869 2/20 0.38
PPARG P37231 1/20 0.38
ACACB O00763 1/20 0.38
ATM Q13315 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA7 P43166 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2573117 0.87 CTSK (0.45) CTSKCTSSTRPA1APPPPARA
SCHEMBL3379781 0.87 CTSK (0.51) CTSKCTSSAPPPPARAPPARG
SCHEMBL844407 0.87 CTSK (0.51) CTSKCTSSAPPPPARAPPARG
SCHEMBL14250689 0.87 CTSK (0.51) CTSKCTSSAPPPPARAPPARG
SCHEMBL4116995 0.87 CTSK (0.51) CTSKCTSSAPPPPARAPPARG
SCHEMBL3414715 0.87 CTSK (0.51) CTSKCTSSAPPPPARAPPARG
SCHEMBL6107389 0.86 CTSK (0.41) CTSKCTSSTRPA1APPPPARA
SCHEMBL22303774 0.86 CTSK (0.41) CTSKCTSSTRPA1APPPPARA
SCHEMBL2436816 0.86 CTSS (0.46) CTSKCTSSTRPA1
SCHEMBL2836398 0.86 TRPA1 (0.52) CTSKCTSSTRPA1PPARAPPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7884204-B2 such as (2S)-2-[(2,6-dichlorobenzoyl)amino]-3-[4-(4-hydroxy-1-methyl-2-oxo-1,2-dihydro-3-quinolinyl)phenyl]propionic acid, used for the teratment of inflammatory diseases, arthritis, inflammatory bowel diseases, lupus, multiple syndrome, asthma, psoriasis, allergies, diabetes and cardiovascular diseases AJINOMOTO CO., INC. (JP) 2011-02-08 US disclosed