Triaziquone

Triaziquone

SCHEMBL1241564

C=C.CC(=O)O.CC(=O)O.CC(=O)O.CC(=O)O.N.N.O=C1C=C(N2CC2)C(=O)C(N2CC2)=C1N1CC1.OB(O)O

nearest known ligand 0.36

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADRA2AADRA2BADRA2CADRB2AGTR1AVPR1AAVPR1BAVPR2BDKRB2CALCRCHRNA3CHRNB4ESR1ESR2GHSRGNRHRGSC1HSPA8MALT1MC1RMC4RNOS1NOS2NOS3OPRK1OXTRRAMP1RAMP2RAMP3SCN5ASSTR1SSTR2SSTR3SSTR4SSTR5dacAdacBdacCfolPftsImrcAmrcBmrdArplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Triaziquone. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.36
MAPT P10636 1/20 0.36
STAT3 P40763 1/20 0.36
HTT P42858 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
DNMT1 P26358 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Triaziquone SCHEMBL10414999 0.92 MAPT (0.41) TP53MAPTSTAT3HTTSMN1; SMN2
Triaziquone SCHEMBL11422311 0.91 MAPT (0.42) TP53MAPTSTAT3HTTSMN1; SMN2
Triaziquone SCHEMBL11744970 0.87 MAPT (0.40) TP53MAPTSTAT3HTTSMN1; SMN2
Triaziquone SCHEMBL1445124 0.84 TP53 (0.38) TP53MAPTSTAT3HTTSMN1; SMN2
Triaziquone SCHEMBL2095563 0.84 TP53 (0.38) TP53MAPTSTAT3HTTSMN1; SMN2
Triaziquone SCHEMBL20359693 0.84 DNMT1 (0.39) TP53MAPTSTAT3HTTSMN1; SMN2
Triaziquone SCHEMBL21805762 0.84 MAPT (0.40) TP53MAPTSTAT3HTTSMN1; SMN2
Triaziquone SCHEMBL4608905 0.84 DNMT1 (0.43) TP53MAPTSTAT3HTTSMN1; SMN2
Triaziquone SCHEMBL8585531 0.83 HTT (0.37) TP53MAPTSTAT3HTTSMN1; SMN2
Triaziquone SCHEMBL10584873 0.82 DNMT1 (0.44) TP53MAPTSTAT3HTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 31 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9441259-B2 Formation of immobilized biological layers for sensing ABBOTT POINT OF CARE INC. (US) 2016-09-13 US disclosed
EP-2225388-B1 COMPOSITIONS FOR FORMING IMMOBILIZED BIOLOGICAL LAYERS FOR SENSING ABBOTT POINT OF CARE INC (US) 2016-03-30 EP disclosed
US-20150275261-A1 FORMATION OF IMMOBILIZED BIOLOGICAL LAYERS FOR SENSING ABBOTT POINT OF CARE INC. (US) 2015-10-01 US disclosed
US-8986526-B2 Formation of immobilized biological layers for sensing ABBOTT POINT OF CARE INC. (US) 2015-03-24 US disclosed
EP-2235513-B1 FORMATION OF IMMOBILIZED BIOLOGICAL LAYERS FOR SENSING ABBOTT POINT OF CARE INC (US) 2014-05-07 EP disclosed
US-20130112558-A1 FORMATION OF IMMOBILIZED BIOLOGICAL LAYERS FOR SENSING ABBOTT POINT OF CARE INC. (US) 2013-05-09 US disclosed
US-8389042-B2 Formation of immobilized biological layers for sensing ABBOTT POINT OF CARE INC. (US) 2013-03-05 US disclosed
US-20120270756-A1 FORMATION OF IMMOBILIZED BIOLOGICAL LAYERS FOR SENSING ABBOTT POINT OF CARE INC. (US) 2012-10-25 US disclosed
US-8268604-B2 Compositions for forming immobilized biological layers for sensing ABBOTT POINT OF CARE INC. (US) 2012-09-18 US disclosed
US-8241697-B2 Formation of immobilized biological layers for sensing ABBOTT POINT OF CARE INC. (US) 2012-08-14 US disclosed
US-20050167269-A1 System for pH-neutral stable electrophoresis gel Life Technologies Corporation 2005-08-04 US disclosed
US-20050167268-A1 System for pH-neutral stable electrophoresis gel Life Technologies Corporation 2005-08-04 US disclosed
US-6783651-B1 System for pH-neutral stable electrophoresis gel INVITROGEN CORPORATION 2004-08-31 US disclosed
US-20030127330-A1 System for pH-neutral stable electrophoresis gel INVITROGEN CORPORATION 2003-07-10 US disclosed
US-20030121784-A1 System for pH-neutral stable electrophoresis gel INVITROGEN CORPORATION 2003-07-03 US disclosed
US-6162338-A System for pH-neutral stable electrophoresis gel NOVEX (US) 2000-12-19 US disclosed
US-6143154-A System for PH-neutral stable electrophoresis gel NOVEX (US) 2000-11-07 US disclosed
US-6096182-A System for pH-neutral stable electrophoresis gel NOVEX (US) 2000-08-01 US disclosed
US-6059948-A System for pH-neutral stable electrophoresis gel NOVEX (US) 2000-05-09 US disclosed
US-5922185-A System for pH-neutral stable electrophoresis gel NOVEL EXPERIMENTAL TECHNOLOGY, INC. (US) 1999-07-13 US disclosed