SCHEMBL1242272

SCHEMBL1242272

NC(=O)CNC(c1ccccc1)C(O)(c1cccnc1)c1cccnc1

nearest known ligand 0.56

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KCNA5 P22460 12/20 0.56
KCNH2 Q12809 7/20 0.47
LMNA P02545 2/20 0.39
EPHX2 P34913 2/20 0.39
HPGD P15428 1/20 0.39
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1243163 0.82 KCNA5 (0.60) KCNA5KCNH2CYP2C9CYP2C19
SCHEMBL1243322 0.81 KCNA5 (0.59) KCNA5KCNH2LMNAHPGDHTT
SCHEMBL9902165 0.80 KCNA5 (0.58) KCNA5KCNH2SMN1; SMN2
SCHEMBL9901968 0.80 KCNA5 (0.58) KCNA5KCNH2SMN1; SMN2
SCHEMBL1242273 0.80 KCNA5 (0.56) KCNA5KCNH2LMNAEPHX2HPGD
SCHEMBL1240478 0.80 KCNA5 (0.55) KCNA5KCNH2SMN1; SMN2CYP2C9CYP2C19
SCHEMBL1242962 0.78 KCNA5 (0.52) KCNA5KCNH2CYP2C9CYP2C19
SCHEMBL4186497 0.78 KCNA5 (0.55) KCNA5KCNH2LMNAEPHX2HPGD
SCHEMBL1243109 0.77 KCNA5 (0.51) KCNA5KCNH2LMNAEPHX2HPGD
SCHEMBL1243112 0.77 KCNA5 (0.51) KCNA5KCNH2LMNAEPHX2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7879839-B2 For treatment and prevention of cardiac arrhythmias; (+-)-2-Morpholin-4-yl-2-phenyl-1,1-dipyridin-3-yl-ethanol; (+-)-2-[(2-methoxyethyl)(methyl)amino]-2-phenyl-1,1-dipyridin-3-ylethanol MERCK SHARP & DOHME CORP. (US) 2011-02-01 US disclosed