SCHEMBL12427265

SCHEMBL12427265

COC1CN(c2cnc3c(NCCO)nc(-c4cnc(N)nc4)nc3c2)C1

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NLRP3 Q96P20 1/20 0.37
MAP3K12 Q12852 2/20 0.34
PIK3CD O00329 10/20 0.34
PIK3CA P42336 10/20 0.34
PIK3CB P42338 10/20 0.34
PIK3CG P48736 10/20 0.34
IRAK1 P51617 1/20 0.33
LATS1 O95835 1/20 0.32
LATS2 Q9NRM7 1/20 0.32
ADORA2A P29274 1/20 0.32
GAK O14976 1/20 0.32
MAPK1 P28482 1/20 0.32
PDE10A Q9Y233 1/20 0.32
APP P05067 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2269892 0.76 PIK3CA (0.57) PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL12427503 0.64 LATS1 (0.37) LATS1LATS2MAPK1
SCHEMBL10239932 0.62 MAP3K12 (0.41) MAP3K12PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL22256141 0.61 TLR8 (0.38) NLRP3GAKMAPK1
SCHEMBL2269763 0.60 PIK3CA (0.59) PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL2272652 0.59 PIK3R1 (0.41) PIK3CDPIK3CAPIK3CBPIK3CGGAK
SCHEMBL4446943 0.58 PIK3CA (0.64) PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL23472667 0.58 TNF (0.49)
SCHEMBL29785073 0.57 EGLN2 (0.35) MAP3K12MAPK1
SCHEMBL14913101 0.57 CHRNB2 (0.42) PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011101429-A1 PYRIDO[3,2-D]PYRIMIDINE PI3K DELTA INHIBITOR COMPOUNDS AND METHODS OF USE F. HOFFMANN-LA ROCHE AG (CH) 2011-08-25 WO disclosed