SCHEMBL12427503

SCHEMBL12427503

Nc1ncc(-c2nc(NCCO)c3nc(OCC(F)(F)F)ccc3n2)cn1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LATS1 O95835 2/20 0.37
LATS2 Q9NRM7 1/20 0.37
MAPK1 P28482 1/20 0.37
SCN9A Q15858 1/20 0.35
ALDH1A1 P00352 2/20 0.35
LMNA P02545 2/20 0.35
HPGD P15428 2/20 0.35
KCNH2 Q12809 1/20 0.35
PTPN1 P18031 1/20 0.34
ALOX5AP P20292 2/20 0.34
FEN1 P39748 2/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
TLR8 Q9NR97 4/20 0.33
TLR7 Q9NYK1 4/20 0.33
TRPV3 Q8NET8 1/20 0.33
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
EPHX2 P34913 1/20 0.32
CYP2J2 P51589 1/20 0.32
PIM1 P11309 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2276345 0.72 PIK3CA (0.60)
SCHEMBL14342919 0.61 PIK3CA (0.49) ALDH1A1CYP2C19TSHR
SCHEMBL29790493 0.59 TLR8 (0.71) MAPK1ALDH1A1TLR8TLR7KDM4E
SCHEMBL17076589 0.59 L3MBTL1 (0.36) MAPK1ALDH1A1L3MBTL1PIM1KDM4E
SCHEMBL18124725 0.59 TLR8 (0.71) MAPK1ALDH1A1TLR8TLR7KDM4E
SCHEMBL22256141 0.58 TLR8 (0.38) MAPK1KCNH2PTPN1TLR8TLR7
SCHEMBL16465803 0.58 NUDT1 (0.41) MAPK1ALDH1A1KCNH2L3MBTL1PIM1
SCHEMBL3159641 0.58 NUDT1 (0.43) MAPK1ALDH1A1PTPN1L3MBTL1CYP2C19
SCHEMBL29625490 0.58 NUDT1 (0.69) ALDH1A1ALOX5APFEN1L3MBTL1PIM1
SCHEMBL29154 0.58 NUDT1 (0.69) ALDH1A1ALOX5APFEN1L3MBTL1PIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011101429-A1 PYRIDO[3,2-D]PYRIMIDINE PI3K DELTA INHIBITOR COMPOUNDS AND METHODS OF USE F. HOFFMANN-LA ROCHE AG (CH) 2011-08-25 WO disclosed