SCHEMBL12428253

SCHEMBL12428253

CC(C)N1CCCC(CCN2CCn3c(c(C4CCCCC4)c4ccc(C(=O)O)cc43)-c3ccc(OCc4ccccc4)cc32)C1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKCA P17252 1/20 0.41
MMP12 P39900 1/20 0.41
NR1I2 O75469 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
MCHR1 Q99705 1/20 0.35
CHRM4 P08173 1/20 0.35
KCNH2 Q12809 2/20 0.34
VDR P11473 2/20 0.34
NR1H4 Q96RI1 2/20 0.34
HRH3 Q9Y5N1 1/20 0.34
CHRNB2 P17787 1/20 0.34
CHRNA5 P30532 1/20 0.34
CHRNA7 P36544 1/20 0.34
CHRNA4 P43681 1/20 0.34
KDM2B Q8NHM5 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12428184 0.92 PRKCA (0.40) PRKCAMMP12NR1I2CYP3A4KCNH2
SCHEMBL12428426 0.91 PRKCA (0.40) PRKCAMMP12NR1I2CYP3A4CYP2C9
SCHEMBL10283247 0.88 PRKCA (0.47) PRKCAMMP12NR1I2CYP3A4CYP2C9
SCHEMBL12428293 0.87 PRKCA (0.41) PRKCAMMP12NR1I2CYP3A4KCNH2
SCHEMBL12427984 0.87 PRKCA (0.42) PRKCAMMP12NR1I2KCNH2
SCHEMBL12428402 0.87 PRKCA (0.42) PRKCAMMP12NR1I2CYP3A4CYP2C9
SCHEMBL12427924 0.86 PRKCA (0.42) PRKCAMMP12NR1I2CYP3A4CYP2C19
SCHEMBL12428182 0.86 PRKCA (0.42) PRKCAMMP12NR1I2CYP3A4CYP2C9
SCHEMBL12428207 0.86 PRKCA (0.40) PRKCAMMP12NR1I2KCNH2
SCHEMBL12428227 0.85 PRKCA (0.41) PRKCAMMP12NR1I2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7977331-B1 Tetracyclic fused heterocyclic compound and use thereof as HCV polymerase inhibitor JAPAN TOBACCO INC. (JP) 2011-07-12 US disclosed
US-7977331-B1 Tetracyclic fused heterocyclic compound and use thereof as HCV polymerase inhibitor JAPAN TOBACCO INC. (JP) 2011-07-12 US disclosed