SCHEMBL12430882

SCHEMBL12430882

CNC(=O)c1ccc2nc(C)[nH]c2c1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.69
ESR2 Q92731 1/20 0.69
TDP1 Q9NUW8 1/20 0.69
POLB P06746 6/20 0.62
ALDH1A1 P00352 5/20 0.62
RAB9A P51151 3/20 0.62
HPGD P15428 3/20 0.62
SMN1; SMN2 Q16637 1/20 0.62
MEN1 O00255 2/20 0.57
KMT2A Q03164 2/20 0.57
NPC1 O15118 1/20 0.57
CHEK2 O96017 3/20 0.55
KDM4E B2RXH2 1/20 0.51
MAPT P10636 1/20 0.51
HDAC6 Q9UBN7 4/20 0.50
HDAC3 O15379 3/20 0.50
HDAC7 Q8WUI4 1/20 0.50
HDAC9 Q9UKV0 1/20 0.50
PLK1 P53350 1/20 0.50
TAS2R8 Q9NYW2 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13306080 0.88 TDP1 (0.53) HSP90AA1ESR2TDP1POLBALDH1A1
SCHEMBL27074031 0.84 HSP90AA1 (0.64) HSP90AA1ESR2TDP1POLBALDH1A1
SCHEMBL9304604 0.83 CHEK2 (0.54) HSP90AA1ESR2TDP1POLBALDH1A1
SCHEMBL6113137 0.82 HSP90AA1 (0.76) HSP90AA1ESR2TDP1POLBALDH1A1
SCHEMBL29924530 0.82 TDP1 (1.00) HSP90AA1ESR2TDP1POLBALDH1A1
SCHEMBL1758956 0.82 TDP1 (1.00) HSP90AA1ESR2TDP1POLBALDH1A1
SCHEMBL4243540 0.81 HSP90AA1 (0.69) HSP90AA1ESR2TDP1POLBALDH1A1
SCHEMBL7428472 0.81 HSP90AA1 (0.73) HSP90AA1ESR2TDP1POLBALDH1A1
Hydrochloric Acid SCHEMBL7331913 0.81 TDP1 (0.97) HSP90AA1ESR2TDP1POLBALDH1A1
SCHEMBL14336559 0.81 ALDH1A1 (0.54) HSP90AA1ESR2TDP1ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024019541-A1 HETEROARYL DERIVATIVE COMPOUND AND USE THEREOF 일동제약(주) 2024-01-25 WO disclosed
EP-1888579-B1 NOVEL FLUORENE DERIVATIVES, COMPOSITION CONTAINING SAID DERIVATIVES AND THE USE THEREOF AVENTIS PHARMA SA (FR) 2011-08-03 EP disclosed