SCHEMBL9304604

SCHEMBL9304604

CNC(=O)c1ccc2nc(S)[nH]c2c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 3/20 0.54
PLK1 P53350 1/20 0.49
HSP90AA1 P07900 1/20 0.48
ESR2 Q92731 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
HDAC6 Q9UBN7 6/20 0.46
HDAC3 O15379 4/20 0.46
HDAC7 Q8WUI4 1/20 0.46
HDAC9 Q9UKV0 1/20 0.46
HDAC1 Q13547 3/20 0.45
HDAC8 Q9BY41 3/20 0.45
HDAC2 Q92769 1/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
AURKA O14965 1/20 0.44
NPY5R Q15761 1/20 0.44
RET P07949 1/20 0.44
ALDH1A1 P00352 2/20 0.44
CCNC P24863 1/20 0.44
CDK8 P49336 1/20 0.44
KDM4E B2RXH2 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9304589 0.88 AURKA (0.47) CHEK2PLK1TDP1HDAC6HDAC8
SCHEMBL12430882 0.83 HSP90AA1 (0.69) CHEK2PLK1HSP90AA1ESR2TDP1
SCHEMBL17821410 0.83 HSP90AA1 (0.51) CHEK2HSP90AA1ESR2TDP1SMN1; SMN2
SCHEMBL6217370 0.82 HTT (0.64) HSP90AA1ESR2TDP1SMN1; SMN2ALDH1A1
SCHEMBL766093 0.81 HSP90AA1 (0.66) CHEK2HSP90AA1ESR2TDP1SMN1; SMN2
SCHEMBL7868231 0.80 CHEK2 (0.60) CHEK2
SCHEMBL29242251 0.80 HSP90AA1 (0.64) CHEK2HSP90AA1ESR2TDP1SMN1; SMN2
SCHEMBL7868225 0.80 HSP90AA1 (0.47) CHEK2HSP90AA1ESR2TDP1SMN1; SMN2
SCHEMBL14336559 0.79 ALDH1A1 (0.54) CHEK2PLK1HSP90AA1ESR2TDP1
SCHEMBL19954465 0.79 CHEK2 (0.52) CHEK2PLK1HSP90AA1ESR2TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5347008-A Thio(cyclo) alkanepolycarboxylic acids containing heterocyclic substituents CIBA-GEIGY CORPORATION (US) 1994-09-13 US disclosed