SCHEMBL12436809

SCHEMBL12436809

CCCOc1cccc(-c2cccnc2)c1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 4/20 0.63
CYP2C9 P11712 2/20 0.63
CYP2C19 P33261 2/20 0.63
CYP3A4 P08684 2/20 0.63
CYP2D6 P10635 1/20 0.63
CYP11B1 P15538 2/20 0.58
CYP11B2 P19099 2/20 0.58
TSHR P16473 1/20 0.54
MAPK1 P28482 1/20 0.54
S1PR1 P21453 1/20 0.53
BACE1 P56817 1/20 0.53
KMT2A Q03164 1/20 0.52
KDM4E B2RXH2 1/20 0.51
FPR2 P25090 1/20 0.51
CYP1A2 P05177 2/20 0.49
CHRNB2 P17787 3/20 0.48
CHRNA4 P43681 2/20 0.48
CYP17A1 P05093 1/20 0.48
EPHX2 P34913 1/20 0.48
PRMT6 Q96LA8 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15740654 0.90 CYP19A1 (0.67) CYP19A1CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL27958859 0.87 CYP19A1 (0.75) CYP19A1CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL4512812 0.87 CYP11B2 (0.79) CYP19A1CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL5749788 0.86 CYP19A1 (0.53) CYP19A1CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL198917 0.85 KDM4E (0.59) CYP19A1CYP2C9CYP2C19TSHRBACE1
SCHEMBL3177161 0.84 MKNK1 (0.56) CYP19A1CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL4865899 0.84 CYP19A1 (0.51) CYP19A1CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL4870398 0.83 CYP19A1 (0.54) CYP19A1CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL171896 0.81 CHRNB2 (0.68) CYP19A1CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL30338591 0.81 CHRNB2 (0.68) CYP19A1CYP2C9CYP2C19CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1802641-B1 BISPHOSPHONATE COMPOUNDS AND METHODS FOR BONE RESORPTION DISEASES, CANCER, BONE PAIN, IMMUNE DISORDERS, AND INFECTIOUS DISEASES UNIV ILLINOIS (US) 2011-08-10 EP disclosed