SCHEMBL12436849

SCHEMBL12436849

CCOc1cc(-c2cccc(C)c2)c2oc(=O)sc2c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 9/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
MAOB P27338 3/20 0.38
ALDH1A1 P00352 5/20 0.37
KDM4E B2RXH2 5/20 0.37
HPGD P15428 3/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
ADORA3 P0DMS8 2/20 0.37
TP53 P04637 1/20 0.37
TSHR P16473 1/20 0.37
MAPK1 P28482 1/20 0.37
CASP3 P42574 1/20 0.37
RAB9A P51151 1/20 0.37
SENP8 Q96LD8 1/20 0.37
HSD17B10 Q99714 1/20 0.37
SENP7 Q9BQF6 1/20 0.37
SENP6 Q9GZR1 1/20 0.37
CA12 O43570 2/20 0.36
CA9 Q16790 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6001485 0.79 MAPT (0.72) MAPTMEN1KMT2AMAOBALDH1A1
SCHEMBL6000138 0.76 KMT2A (0.44) MAPTMEN1KMT2AMAOBALDH1A1
SCHEMBL12225772 0.67 RXRA (0.57) MAPTALDH1A1KDM4EHPGDSMN1; SMN2
SCHEMBL10104745 0.67 ALDH1A1 (0.53) MAPTKMT2AMAOBALDH1A1KDM4E
SCHEMBL23309025 0.66 FFAR1 (0.49) MAPTALDH1A1KDM4EHPGDSMN1; SMN2
SCHEMBL2623677 0.65 NQO1 (0.52) ALDH1A1KDM4EHPGDSMN1; SMN2TP53
SCHEMBL12436603 0.64 KMT2A (0.46) MAPTMEN1KMT2AALDH1A1KDM4E
SCHEMBL2129509 0.64 MAOA (0.66) MAPTMEN1KMT2AMAOBALDH1A1
SCHEMBL6000106 0.64 MAPT (0.77) MAPTMEN1KMT2AMAOBALDH1A1
SCHEMBL15503719 0.63 MAPT (1.00) MAPTMEN1KMT2AMAOBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011094708-A2 SMALL MOLECULES FOR THE MODULATION OF MCL-1 AND METHODS OF MODULATIING CELL DEATH, CELL DIVISION, CELL DIFFERENTIATION AND METHODS OF TREATING DISORDERS DANA-FARBER CANCER INSTITUTE, INC (US) 2011-08-04 WO disclosed