SCHEMBL12436906

SCHEMBL12436906

COC(=O)NCC1(C(C)=O)CCOCC1

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.35
ALDH1A1 P00352 5/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
POLB P06746 1/20 0.32
P2RX7 Q99572 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
LMNA P02545 1/20 0.31
EPHX1 P07099 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
PKM P14618 1/20 0.31
CYP2C19 P33261 1/20 0.31
HTR2A P28223 1/20 0.30
SLC6A5 Q9Y345 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12436899 0.84 HCRTR2 (0.44) TSHRALDH1A1L3MBTL1SMN1; SMN2EPHX1
SCHEMBL12436902 0.84 OPRM1 (0.33) TSHRALDH1A1L3MBTL1P2RX7
SCHEMBL12436903 0.72 ALDH1A1 (0.57) ALDH1A1L3MBTL1POLBP2RX7SMN1; SMN2
SCHEMBL13804310 0.71 SMN1; SMN2 (0.32) SMN1; SMN2EPHX1
SCHEMBL1970278 0.71 HCRTR2 (0.44) TSHRALDH1A1SMN1; SMN2EPHX1
SCHEMBL16076549 0.70 TDP1 (0.46) TSHRALDH1A1EPHX1
SCHEMBL16038053 0.70 HCRTR2 (0.43) TSHRALDH1A1L3MBTL1SMN1; SMN2EPHX1
SCHEMBL16391319 0.70 TSHR (0.33) TSHR
SCHEMBL12587392 0.70 SMN1; SMN2 (0.31) SMN1; SMN2
SCHEMBL14811020 0.69 ACHE (0.44) ALDH1A1POLBSMN1; SMN2LMNACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE49686-E1 Nitrogen-containing heterocyclic compound and use of same TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2023-10-10 US disclosed
US-RE49686-E1 Nitrogen-containing heterocyclic compound and use of same TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2023-10-10 US disclosed
US-RE48334-E1 Nitrogen-containing heterocyclic compound and use of same TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2020-12-01 US disclosed
US-20110178060-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND AND USE OF SAME TAKEDA PHARMACEUTICAL COMPANY LIMITED 2011-07-21 US disclosed
US-20110178060-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND AND USE OF SAME TAKEDA PHARMACEUTICAL COMPANY LIMITED 2011-07-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110178060-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND AND USE OF SAME NTSR2, BDKRB1, AVPR1B TSHR 183/4885ALDH1A1 3648/4885L3MBTL1 1003/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.