SCHEMBL12439655

SCHEMBL12439655

CCCc1cc2nc(-c3cc(C)nn3C)oc2cc1CCC

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 4/20 0.40
KCNH2 Q12809 4/20 0.40
ADORA2B P29275 1/20 0.34
F2RL3 Q96RI0 2/20 0.33
ESR1 P03372 1/20 0.32
ESR2 Q92731 1/20 0.32
KDM4E B2RXH2 2/20 0.31
NPC1 O15118 2/20 0.31
ALDH1A1 P00352 2/20 0.31
HPGD P15428 2/20 0.31
RAB9A P51151 2/20 0.31
SMN1; SMN2 Q16637 2/20 0.31
HSD17B10 Q99714 2/20 0.31
MAPT P10636 1/20 0.31
HRH1 P35367 1/20 0.31
TP53 P04637 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2310141 0.72 DRD3 (0.49) DRD3KCNH2HRH1
SCHEMBL10126049 0.65 ESR1 (0.44) ESR1ESR2KDM4ENPC1ALDH1A1
SCHEMBL13621036 0.64 SMN1; SMN2 (0.47) ESR1ESR2KDM4ENPC1ALDH1A1
SCHEMBL26827234 0.63 HSD17B10 (0.50) F2RL3KDM4ENPC1ALDH1A1HPGD
SCHEMBL16487535 0.63 SMN1; SMN2 (0.42) ADORA2BKDM4ENPC1ALDH1A1HPGD
SCHEMBL20757447 0.61 ADORA2B (0.32) KCNH2ADORA2BMEN1KMT2A
SCHEMBL10077232 0.61 MEN1 (0.40) KCNH2SMN1; SMN2MEN1KMT2A
SCHEMBL12440017 0.60 LMNA (0.35) DRD3ALDH1A1
SCHEMBL12072250 0.59 S1PR1 (0.39) ADORA2BKDM4EALDH1A1MAPT
SCHEMBL3523330 0.58 NOTUM (0.50) KDM4EALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1751163-B1 BENZAZEPINE COMPOUNDS HAVING AFFINITY FOR DOPAMINE D3 RECEPTOR AND USES THEREOF GLAXO GROUP LTD (GB) 2011-08-10 EP disclosed