SCHEMBL12439725

SCHEMBL12439725

CCN(CCN(C)C(=O)OC(C)(C)C)CCn1cc(-c2cncc(-c3cc(-c4cc(Cl)ccc4F)nc4ncccc34)c2)cn1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACACB O00763 1/20 0.34
ACACA Q13085 1/20 0.34
TGFBR1 P36897 5/20 0.33
MAP4K4 O95819 2/20 0.33
ACVR1B P36896 2/20 0.32
ACVRL1 P37023 2/20 0.32
KAT6A Q92794 1/20 0.31
KAT5 Q92993 1/20 0.31
HTR1A P08908 1/20 0.31
DRD3 P35462 1/20 0.31
OPRK1 P41145 1/20 0.31
HTR3A P46098 1/20 0.31
KCNH2 Q12809 1/20 0.31
GHSR Q92847 1/20 0.31
HTR2C P28335 1/20 0.31
SLC6A4 P31645 1/20 0.31
MET P08581 1/20 0.31
SYK P43405 1/20 0.30
IDO1 P14902 1/20 0.30
SCN9A Q15858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12440840 0.94 ACACB (0.37) ACACBACACATGFBR1MAP4K4ACVR1B
SCHEMBL12439726 0.88 TGFBR1 (0.41) TGFBR1MAP4K4HTR1ADRD3OPRK1
SCHEMBL12440047 0.82 TGFBR1 (0.46) TGFBR1MAP4K4METIDO1
SCHEMBL13968476 0.80 CYP3A4 (0.41)
SCHEMBL2325058 0.80 TGFBR1 (0.41) TGFBR1MAP4K4METIDO1
SCHEMBL2327513 0.79 MET (0.42) TGFBR1METPDK2
SCHEMBL12440044 0.78 FEN1 (0.43) TGFBR1MAP4K4MAPK1
SCHEMBL12440841 0.77 TGFBR1 (0.36) TGFBR1MAP4K4METIDO1MAPK1
SCHEMBL13968445 0.76 TGFBR1 (0.45) TGFBR1MAP4K4METHCRTR1HCRTR2
SCHEMBL13968474 0.75 KDR (0.36) TGFBR1MAP4K4ACVRL1METMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011095196-A1 HETARYL-[1,8]NAPHTHYRIDINE DERIVATIVES MERCK PATENT GMBH (DE) 2011-08-11 WO disclosed