SCHEMBL12445340

SCHEMBL12445340

C(\CN1CCC[C@H](c2ccccc2)C1)=C1\CCCc2c1cnn2-c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 3/20 0.42
DRD3 P35462 3/20 0.42
DRD4 P21917 2/20 0.42
DRD1 P21728 1/20 0.42
DRD5 P21918 1/20 0.42
SIGMAR1 Q99720 2/20 0.39
TMEM97 Q5BJF2 1/20 0.39
CA1 P00915 2/20 0.36
CA2 P00918 2/20 0.36
CA4 P22748 2/20 0.36
CA9 Q16790 2/20 0.36
HTR7 P34969 1/20 0.36
CNR2 P34972 1/20 0.36
USP30 Q70CQ3 1/20 0.36
HSD11B1 P28845 1/20 0.36
KEAP1 Q14145 1/20 0.36
NFE2L2 Q16236 1/20 0.36
TP53 P04637 2/20 0.35
KDM4E B2RXH2 1/20 0.34
NPC1 O15118 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL956945 1.00 DRD2 (0.42) DRD2DRD3DRD4DRD1DRD5
SCHEMBL956948 1.00 DRD2 (0.42) DRD2DRD3DRD4DRD1DRD5
SCHEMBL956947 1.00 DRD2 (0.42) DRD2DRD3DRD4DRD1DRD5
SCHEMBL955505 0.96 SIGMAR1 (0.39) DRD2DRD3DRD4DRD1DRD5
SCHEMBL955506 0.96 SIGMAR1 (0.39) DRD2DRD3DRD4DRD1DRD5
SCHEMBL955504 0.96 SIGMAR1 (0.39) DRD2DRD3DRD4DRD1DRD5
Oxalic Acid SCHEMBL955889 0.93 KEAP1 (0.39) DRD2DRD3DRD4DRD1DRD5
Oxalic Acid SCHEMBL955891 0.93 KEAP1 (0.39) DRD2DRD3DRD4DRD1DRD5
SCHEMBL959515 0.91 DRD2 (0.42) DRD2DRD3DRD4SIGMAR1TMEM97
SCHEMBL959513 0.91 DRD2 (0.42) DRD2DRD3DRD4SIGMAR1TMEM97

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1781619-B1 SIGMA RECEPTOR INHIBITORS ESTEVE LABOR DR (ES) 2011-08-17 EP disclosed