SCHEMBL12445903

SCHEMBL12445903

Bc1ccc(-c2cc(F)cc(F)c2)c(F)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 1/20 0.39
PDE3A Q14432 1/20 0.39
ESR1 P03372 2/20 0.33
ESR2 Q92731 2/20 0.33
TTR P02766 2/20 0.33
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
USP2 O75604 1/20 0.32
ALDH1A1 P00352 1/20 0.32
DHFR P00374 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
LMNA P02545 1/20 0.32
ALB P02768 1/20 0.32
HMGB1 P09429 1/20 0.32
HPGD P15428 1/20 0.32
CXCL12 P48061 1/20 0.32
KMT2A Q03164 1/20 0.32
HIF1A Q16665 1/20 0.32
SLC22A6 Q4U2R8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL257632 0.83 APP (0.41) PDE3BPDE3AESR1ESR2TTR
SCHEMBL19993198 0.80 ESR1 (0.38) ESR1ESR2TTRKDM4EMEN1
SCHEMBL14926554 0.79 TTR (0.46) PDE3BPDE3AESR1ESR2TTR
SCHEMBL16104369 0.78 LMNA (0.46) PDE3BPDE3AESR1MEN1LMNA
SCHEMBL19993062 0.78 ESR1 (0.41) PDE3BPDE3AESR1ESR2TTR
SCHEMBL30665731 0.74 ALOX5AP (0.45) PDE3BPDE3AESR1ESR2TTR
SCHEMBL29097482 0.74 AHR (0.42) PDE3BPDE3AKDM4E
SCHEMBL12198995 0.74 ALOX5AP (0.45) PDE3BPDE3AESR1ESR2TTR
SCHEMBL12357201 0.74 CTSA (0.44) PDE3BPDE3AMEN1ALDH1A1HPGD
SCHEMBL2246071 0.74 ESR1 (0.60) ESR1ESR2CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3071669-B1 MESOGENIC MEDIA AND LIQUID CRYSTAL DISPLAY DEVICE MERCK PATENT GMBH (DE) 2018-06-20 EP disclosed
EP-2729549-B1 BIMESOGENIC COMPOUNDS MERCK PATENT GMBH (DE) 2016-12-07 EP disclosed
WO-2013004333-A1 BIMESOGENIC COMPOUNDS MERCK PATENT GMBH (DE) 2013-01-10 WO disclosed
EP-2360229-A1 OPTICALLY ISOTROPIC LIQUID CRYSTAL MEDIUM AND OPTICAL ELEMENT JNC Corporation (JP) 2011-08-24 EP disclosed