SCHEMBL12458971

SCHEMBL12458971

CC(O)(CNC(=O)Nc1ccc(OC2CCN(Cc3ccc(C(C)(O)C(F)(F)F)cc3)C2)cc1)C(F)(F)F

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 3/20 0.45
CHRM4 P08173 1/20 0.43
CCR3 P51677 1/20 0.43
DNMT1 P26358 1/20 0.43
EHMT2 Q96KQ7 1/20 0.43
TP53 P04637 2/20 0.42
PRKAB2 O43741 2/20 0.41
PRKAG1 P54619 2/20 0.41
PRKAA2 P54646 2/20 0.41
PRKAA1 Q13131 2/20 0.41
PRKAG3 Q9UGI9 2/20 0.41
PRKAG2 Q9UGJ0 2/20 0.41
PRKAB1 Q9Y478 2/20 0.41
KCNH2 Q12809 1/20 0.40
GPR119 Q8TDV5 1/20 0.40
MCHR1 Q99705 1/20 0.40
FAAH O00519 1/20 0.40
UTS2R Q9UKP6 1/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12273956 0.94 ADRB2 (0.45) ADRB2CHRM4CCR3DNMT1EHMT2
SCHEMBL12458970 0.90 TP53 (0.50) ADRB2CHRM4CCR3DNMT1EHMT2
SCHEMBL1867375 0.84 ADRB2 (0.49) ADRB2CHRM4DNMT1EHMT2PRKAB2
SCHEMBL12274902 0.82 TP53 (0.50) ADRB2CHRM4CCR3DNMT1EHMT2
SCHEMBL17010808 0.79 TP53 (0.47) ADRB2CHRM4CCR3DNMT1EHMT2
SCHEMBL15493055 0.79 FLT3 (0.46) ADRB2DNMT1EHMT2PRKAB2PRKAG1
SCHEMBL17010810 0.78 CCR3 (0.42) ADRB2CHRM4CCR3DNMT1EHMT2
SCHEMBL12274653 0.78 ADRB2 (0.50) ADRB2CHRM4DNMT1EHMT2TP53
SCHEMBL12524264 0.78 ADRB2 (0.48) ADRB2CHRM4DNMT1EHMT2PRKAB2
SCHEMBL1868406 0.75 ADRB2 (0.53) ADRB2DNMT1EHMT2PRKAB2PRKAG1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9108939-B2 (1, 1, 1,3,3,3-hexafluoro-2 hydroxypropan-2-yl) phenyl derivative, pharmaceutical compositions thereof and their use for the treatment of atherosclerosis MERCK SHARP & DOHME B.V. (NL) 2015-08-18 US disclosed
US-20120238574-A1 (1, 1, 1,3,3,3 -HEXAFLUORO-2 HYDROXYPROPAN- 2 -YL) PHENYL DERIVATIVE, PHARMACEUTICAL COMPOSITIONS THEREOF AND THEIR USE FOR THE TREATMENT OF ATHEROSCLEROSIS N.V. ORGANON (NL) 2012-09-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120238574-A1 (1, 1, 1,3,3,3 -HEXAFLUORO-2 HYDROXYPROPAN- 2 -YL) PHENYL DERIVATIVE, PHARMACEUTICAL COMPOSITIONS THEREOF AND THEIR USE FOR THE TREATMENT OF ATHEROSCLEROSIS TGFB1, FPR1, TGFB2 ADRB2 120/4885CHRM4 2919/4885CCR3 1208/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.