SCHEMBL12459652

SCHEMBL12459652

Nc1ccc(C(=O)NCc2ncc[nH]2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.52
FPR2 P25090 1/20 0.49
KDM4E B2RXH2 2/20 0.47
NAMPT P43490 2/20 0.47
MAPT P10636 1/20 0.47
HIF1A Q16665 1/20 0.47
SLC22A6 Q4U2R8 1/20 0.47
SLC22A8 Q8TCC7 1/20 0.47
ADORA3 P0DMS8 1/20 0.47
ADORA2A P29274 1/20 0.47
ADORA2B P29275 1/20 0.47
ADORA1 P30542 1/20 0.47
KLK1 P06870 1/20 0.47
KLK5 Q9Y337 1/20 0.47
EPHX2 P34913 1/20 0.47
GAA P10253 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
LMNA P02545 3/20 0.44
MAPK1 P28482 2/20 0.44
SLC22A2 O15244 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14817907 0.85 ROCK2 (0.52) ROCK2FPR2KDM4ENAMPTMAPT
SCHEMBL31188529 0.85 GAA (0.60) ROCK2FPR2KDM4EMAPTGAA
SCHEMBL7011089 0.83 NAMPT (0.65) NAMPT
SCHEMBL18617522 0.83 ROCK2 (0.50) ROCK2FPR2NAMPTADORA3ADORA2A
SCHEMBL20671963 0.82 ROCK2 (0.47) ROCK2FPR2MAPTADORA3ADORA2A
SCHEMBL3769508 0.82 ROCK2 (0.49) ROCK2FPR2KDM4ENAMPTADORA3
SCHEMBL21335657 0.81 PLK1 (0.50) ROCK2FPR2KDM4ENAMPTADORA3
SCHEMBL31680532 0.81 TAAR1 (0.55) ROCK2FPR2KDM4ENAMPTMAPT
SCHEMBL6451096 0.77 FPR2 (0.55) ROCK2FPR2KDM4EADORA3ADORA2A
SCHEMBL1258259 0.76 FPR2 (0.54) ROCK2FPR2ADORA3ADORA2AADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2343303-A1 PI3-kinase inhibitors Boehringer Ingelheim International GmbH (DE) 2011-07-13 EP disclosed