SCHEMBL14817907

SCHEMBL14817907

Cc1ccc(C(=O)NCc2ncc[nH]2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.52
NPC1 O15118 3/20 0.51
RAB9A P51151 2/20 0.51
SMN1; SMN2 Q16637 3/20 0.49
HTT P42858 2/20 0.49
MMP13 P45452 2/20 0.49
FPR2 P25090 1/20 0.49
MMP2 P08253 1/20 0.49
CYP3A4 P08684 1/20 0.49
STAT3 P40763 1/20 0.49
MAPK14 Q16539 1/20 0.49
NAMPT P43490 1/20 0.47
ADORA3 P0DMS8 1/20 0.47
ADORA2A P29274 1/20 0.47
ADORA2B P29275 1/20 0.47
ADORA1 P30542 1/20 0.47
MAPT P10636 3/20 0.47
ALDH1A1 P00352 2/20 0.47
TDP1 Q9NUW8 2/20 0.47
POLB P06746 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18617522 0.86 ROCK2 (0.50) ROCK2SMN1; SMN2FPR2NAMPTADORA3
SCHEMBL12459652 0.85 ROCK2 (0.52) ROCK2NPC1RAB9ASMN1; SMN2HTT
SCHEMBL31188529 0.85 GAA (0.60) ROCK2NPC1RAB9ASMN1; SMN2HTT
SCHEMBL21335657 0.83 PLK1 (0.50) ROCK2SMN1; SMN2FPR2NAMPTADORA3
SCHEMBL20671963 0.82 ROCK2 (0.47) ROCK2NPC1RAB9ASMN1; SMN2HTT
SCHEMBL3769508 0.82 ROCK2 (0.49) ROCK2SMN1; SMN2HTTFPR2NAMPT
SCHEMBL18735743 0.82 KLK1 (0.50) ROCK2NPC1RAB9AFPR2NAMPT
SCHEMBL31680532 0.81 TAAR1 (0.55) ROCK2NPC1RAB9ASMN1; SMN2HTT
SCHEMBL6451096 0.77 FPR2 (0.55) ROCK2SMN1; SMN2HTTFPR2ADORA3
SCHEMBL5630316 0.76 FPR2 (0.54) ROCK2SMN1; SMN2FPR2ADORA3ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1802636-B1 PI3 KINASES INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2013-03-27 EP disclosed