SCHEMBL12463147

SCHEMBL12463147

CSc1cnc(Cl)nc1NCCO

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.42
KDM4E B2RXH2 3/20 0.41
MAPK1 P28482 2/20 0.41
FLT3 P36888 2/20 0.38
PLK4 O00444 1/20 0.38
AURKA O14965 1/20 0.38
DCLK1 O15075 1/20 0.38
ROCK2 O75116 1/20 0.38
PRKD3 O94806 1/20 0.38
MAP4K4 O95819 1/20 0.38
CDK1 P06493 1/20 0.38
FES P07332 1/20 0.38
ROS1 P08922 1/20 0.38
FGFR1 P11362 1/20 0.38
PHKG2 P15735 1/20 0.38
PRKACA P17612 1/20 0.38
FLT1 P17948 1/20 0.38
RPS6KB1 P23443 1/20 0.38
CDK2 P24941 1/20 0.38
MARK3 P27448 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1917420 0.81 GLP1R (0.46) KDM4EMAPK1CLK4IRAK4STK17B
SCHEMBL14112779 0.79 KDM4E (0.45) HTTKDM4EMAPK1STK17BSTK17A
SCHEMBL1938460 0.78 STK17A (0.51) HTTKDM4EMAPK1STK17BSTK17A
SCHEMBL5419429 0.76 XDH (0.39) KDM4EALDH1A1KMT2AL3MBTL1MEN1
SCHEMBL11908962 0.76 ALDH1A1 (0.59) HTTKDM4EMAPK1STK17BSTK17A
SCHEMBL2817011 0.76 HTT (0.41) HTTKDM4EMAPK1STK17BSTK17A
SCHEMBL1774700 0.76 KMT2A (0.43) HTTKDM4EMAPK1STK17BSTK17A
SCHEMBL25902572 0.75 HTT (0.58) HTTKDM4EMAPK1STK17BSTK17A
SCHEMBL25902576 0.73 HTT (0.40) HTTKDM4EMAPK1STK17BSTK17A
SCHEMBL27502303 0.72 CSNK1A1 (0.51) HTTKDM4EMAPK1AURKACDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011080568-A2 NOVEL PYRIMIDINE COMPOUNDS AS MTOR AND P13K INHIBITORS DEVELOPMENT CENTER FOR BIOTECHNOLOGY (TW) 2011-07-07 WO disclosed