SCHEMBL12464484

SCHEMBL12464484

Cc1cc(C[C@H](N)C(=O)N[C@H](Cc2ccc(I)cc2)C(=O)N[C@H](Cc2ccccc2)C(=O)N[C@H](Cc2c[nH]c3ccccc23)C(N)=O)ccc1O

nearest known ligand 0.60

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CCKAR P32238 2/20 0.56
CCKBR P32239 2/20 0.56
OPRM1 P35372 1/20 0.55
OPRD1 P41143 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12464294 0.89 OPRM1 (0.57) OPRM1OPRD1
SCHEMBL12464360 0.85 NPY1R (0.56)
SCHEMBL13725698 0.84 ECE1 (0.64)
SCHEMBL22133113 0.84 ECE1 (0.64)
SCHEMBL30799684 0.84 ECE1 (0.64)
SCHEMBL29966716 0.83 OPRM1 (0.72) OPRM1OPRD1
SCHEMBL12464361 0.82 CTSC (0.53)
SCHEMBL12464362 0.82
SCHEMBL31722484 0.82 KDM4E (0.62)
SCHEMBL29966936 0.81 GHSR (0.67) OPRM1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110183358-A1 METHODS AND COMPOSITIONS FOR DEREPRESSION OF IAP-INHIBITED CASPASE THE BURNHAM INSTITUTE (US) 2011-07-28 US disclosed