SCHEMBL124646

SCHEMBL124646

CC(C)(C)OC(=O)N1CCC(CNS(C)(=O)=O)CC1

nearest known ligand 0.55

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 13/20 0.55
KDM4E B2RXH2 2/20 0.55
PKM P14618 1/20 0.55
GPR119 Q8TDV5 4/20 0.51
MAPT P10636 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21194508 0.92 TGFBR1 (0.48) TGFBR1KDM4EPKMGPR119MAPT
SCHEMBL29160799 0.87 TGFBR1 (0.54) TGFBR1KDM4EPKMGPR119MAPT
SCHEMBL20771440 0.87 KDM4E (0.57) TGFBR1KDM4EPKMGPR119MAPT
SCHEMBL23003379 0.85 NAMPT (0.51) TGFBR1KDM4EPKMGPR119
SCHEMBL26665931 0.85 TGFBR1 (0.53) TGFBR1KDM4EPKMGPR119MAPT
SCHEMBL6402117 0.85 TGFBR1 (0.53) TGFBR1KDM4EPKMGPR119MAPT
SCHEMBL5573225 0.85 KDM4E (0.63) TGFBR1KDM4EPKMGPR119
SCHEMBL21664401 0.84 SCN9A (0.52) TGFBR1MAPT
SCHEMBL372033 0.82 NR1H2 (0.54) KDM4EPKMGPR119
SCHEMBL627965 0.82 KDM4E (0.60) TGFBR1KDM4EPKMGPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230340011-A1 STEROIDAL COMPOSITIONS AND METHODS OF TREATING LIPOGENIC CANCERS Asteroid Therapeutics 2023-10-26 US disclosed
US-20230340011-A1 STEROIDAL COMPOSITIONS AND METHODS OF TREATING LIPOGENIC CANCERS Asteroid Therapeutics 2023-10-26 US disclosed
EP-2201002-B1 5-HT7 RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2012-03-07 EP disclosed
US-7910588-B2 5-HT7 receptor antagonists ELI LILLY AND COMPANY (US) 2011-03-22 US disclosed
US-20100197700-A1 5-HT7 RECEPTOR ANTAGONISTS ELI LILLY AND COMPANY 2010-08-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100197700-A1 5-HT7 RECEPTOR ANTAGONISTS HTR7, HTR1A, HTR2C TGFBR1 1225/4885KDM4E 2286/4885PKM 3252/4885
US-20230340011-A1 STEROIDAL COMPOSITIONS AND METHODS OF TREATING LIPOGENIC CANCERS SREBF1, SREBF2, NR1H3 TGFBR1 2309/4885KDM4E 2203/4885PKM 2772/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.