SCHEMBL12464650

SCHEMBL12464650

Cc1ccc(CN(C(=O)C(C)C)c2csc(-c3ccccc3)c2)cc1

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 9/20 0.50
LTB4R2 Q9NPC1 1/20 0.49
TSPO P30536 1/20 0.40
HTT P42858 2/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
CNR2 P34972 1/20 0.40
PTGES O14684 1/20 0.39
ALOX5 P09917 1/20 0.39
NPC1 O15118 1/20 0.39
JAK2 O60674 1/20 0.39
ALDH1A1 P00352 1/20 0.39
RAB9A P51151 1/20 0.39
PAX8 Q06710 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2157845 0.90 LTB4R2 (0.48) NR1H4LTB4R2KMT2A
SCHEMBL2157679 0.90 NR1H4 (0.47) NR1H4LTB4R2TSPOHTTMEN1
SCHEMBL2158067 0.88 NR1H4 (0.52) NR1H4LTB4R2MEN1KMT2APTGES
SCHEMBL12464572 0.87 LTB4R2 (0.46) NR1H4LTB4R2PTGES
SCHEMBL2158851 0.85 LTB4R2 (0.48) LTB4R2TSPOHTTMEN1KMT2A
SCHEMBL12464236 0.82 CPB1 (0.51) NR1H4TSPOHTTMEN1KMT2A
SCHEMBL2158539 0.81 ALDH1A1 (0.41) NR1H4LTB4R2ALDH1A1
SCHEMBL2158059 0.79 RIPK1 (0.40) NR1H4LTB4R2MEN1KMT2AALDH1A1
SCHEMBL2158746 0.79 LTB4R2 (0.52) LTB4R2TSPOHTTMEN1KMT2A
SCHEMBL3812537 0.77 LTB4R2 (0.45) NR1H4LTB4R2MEN1KMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7985769-B2 Compounds and methods for the treatment or prevention of Flavivirus infections VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-07-26 US disclosed