SCHEMBL1246560

SCHEMBL1246560

NCc1cccc(S(=O)(=O)NCCNC(=O)O)c1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.51
AKR1C3 P42330 4/20 0.51
USP2 O75604 1/20 0.51
TPSAB1 Q15661 2/20 0.50
PRMT1 Q99873 1/20 0.50
ALDH1A1 P00352 1/20 0.50
HTR6 P50406 1/20 0.49
CYP2C19 P33261 2/20 0.49
CYP1A2 P05177 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49
TSHR P16473 1/20 0.49
HDAC2 Q92769 1/20 0.48
HDAC8 Q9BY41 1/20 0.48
HDAC6 Q9UBN7 1/20 0.48
HTT P42858 1/20 0.47
ATM Q13315 1/20 0.47
MAPK1 P28482 1/20 0.46
TDP1 Q9NUW8 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12407044 0.82 CYP2C19 (0.60) KMT2AAKR1C3TPSAB1PRMT1ALDH1A1
SCHEMBL13637021 0.82 PRMT1 (0.54) KMT2AAKR1C3TPSAB1PRMT1ALDH1A1
SCHEMBL1246677 0.81 CA2 (0.48) KMT2AAKR1C3USP2
Hydrochloric Acid SCHEMBL4636067 0.81 CYP2C19 (0.58) KMT2AAKR1C3TPSAB1PRMT1ALDH1A1
SCHEMBL21051622 0.80 USP2 (0.68) KMT2AUSP2ALDH1A1MAPK1TDP1
SCHEMBL18498633 0.80 ATM (0.72) KMT2AAKR1C3USP2ALDH1A1CYP2C19
SCHEMBL4615322 0.78 KEAP1 (0.69) PRMT1ALDH1A1HTR6CYP1A2HDAC2
SCHEMBL1246685 0.77 SCN9A (0.52) KMT2AAKR1C3USP2ALDH1A1CYP2C19
Hydrochloric Acid SCHEMBL4010772 0.77 KEAP1 (0.67) PRMT1ALDH1A1HTR6CYP1A2HDAC2
SCHEMBL4615715 0.76 HTR6 (0.53) KMT2ATPSAB1PRMT1ALDH1A1HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2286221-A2 METHODS FOR ASSAYING COMPOUNDS OR AGENTS FOR ABILITY TO DISPLACE POTENT LIGANDS OF HEMATOPOIETIC PROSTAGLANDIN D SYNTHASE Cayman Chemical Company (US) 2011-02-23 EP disclosed
WO-2009140364-A2 METHODS FOR ASSAYING COMPOUNDS OR AGENTS FOR ABILITY TO DISPLACE POTENT LIGANDS OF HEMATOPOIETIC PROSTAGLANDIN D SYNTHASE CAYMAN CHEMICAL COMPANY (US) 2009-11-19 WO disclosed