SCHEMBL12465773

SCHEMBL12465773

Nc1cc(-c2cccc(C(F)(F)F)c2)cs1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.48
TSHR P16473 1/20 0.48
MAOB P27338 1/20 0.46
KDM1A O60341 1/20 0.45
KIF11 P52732 1/20 0.44
ALDH1A1 P00352 2/20 0.44
ADORA2A P29274 2/20 0.43
ADORA1 P30542 2/20 0.43
IKBKB O14920 1/20 0.43
BRD4 O60885 1/20 0.43
XDH P47989 1/20 0.42
LTA4H P09960 1/20 0.42
NOTUM Q6P988 2/20 0.41
IDO1 P14902 1/20 0.41
GAA P10253 1/20 0.40
RAB9A P51151 1/20 0.40
RORB Q92753 1/20 0.40
AR P10275 1/20 0.40
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL12465871 0.98 MAOB (0.49) MAPK1TSHRMAOBKDM1AKIF11
SCHEMBL1263144 0.79 TSHR (0.58) MAPK1TSHRMAOBKDM1AKIF11
SCHEMBL29678302 0.79 TSHR (0.58) MAPK1TSHRMAOBKDM1AKIF11
Ammonia Solution, Strong SCHEMBL20472961 0.77 MAOB (0.56) MAPK1TSHRMAOBKDM1AKIF11
SCHEMBL3789224 0.76 TSHR (0.76) MAPK1TSHRMAOBKDM1AKIF11
Hydrochloric Acid SCHEMBL12465771 0.75 TAAR1 (0.53) ALDH1A1ADORA2ANOTUMKDM4EMEN1
SCHEMBL3793159 0.74 MAOB (0.65) MAPK1TSHRMAOBKDM1AKIF11
SCHEMBL24342416 0.74 TSHR (0.50) MAPK1TSHRMAOBKDM1AKIF11
SCHEMBL474410 0.73 LTA4H (0.67) ALDH1A1XDHLTA4HRAB9AAR
SCHEMBL307920 0.73 KIF11 (0.62) MAPK1TSHRMAOBKDM1AKIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012100732-A1 RETINOID-RELATED ORPHAN RECEPTOR GAMMA MODULATORS, COMPOSITION CONTAINING THEM AND USES THEREOF GLAXO GROUP LIMITED (GB) 2012-08-02 WO disclosed