SCHEMBL12465779

SCHEMBL12465779

CC(C)CP(CC(C)C)c1ccccc1-c1ccccc1N(C)C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.38
MAPT P10636 3/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
NSD2 O96028 1/20 0.38
EGFR P00533 1/20 0.38
LMNA P02545 1/20 0.38
MAPK1 P28482 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
MEN1 O00255 1/20 0.31
RAB9A P51151 1/20 0.31
KMT2A Q03164 1/20 0.31
PTK2B Q14289 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
SMN1; SMN2 Q16637 2/20 0.31
KCNN4 O15554 1/20 0.31
TP53 P04637 1/20 0.31
GAA P10253 1/20 0.31
TSHR P16473 1/20 0.31
HTT P42858 1/20 0.30
HIF1A Q16665 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14809988 0.86 CYBB (0.33) ALDH1A1MAPK1MEN1KMT2ASMN1; SMN2
SCHEMBL14820737 0.77 ALDH1A1 (0.41) ALDH1A1MAPTL3MBTL1NSD2EGFR
SCHEMBL7930351 0.75 ALDH1A1 (0.33) ALDH1A1MAPTL3MBTL1NSD2EGFR
SCHEMBL7088869 0.75 TAAR1 (0.31) ALDH1A1L3MBTL1TDP1SMN1; SMN2TSHR
SCHEMBL4717661 0.75 DPP4 (0.35) ALDH1A1MAPTMAPK1KMT2ANPSR1
SCHEMBL2919461 0.73 MAPT (0.52) ALDH1A1MAPTL3MBTL1NSD2EGFR
SCHEMBL29406125 0.70 MAPT (0.37) ALDH1A1MAPTL3MBTL1NSD2EGFR
SCHEMBL29822698 0.70 ALDH1A1 (0.41) ALDH1A1MAPTL3MBTL1NSD2EGFR
SCHEMBL229536 0.70 ALDH1A1 (0.41) ALDH1A1MAPTL3MBTL1NSD2EGFR
SCHEMBL238097 0.70 MAPT (0.37) ALDH1A1MAPTL3MBTL1NSD2EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2668165-A1 NOVEL TETRAHYDROQUINOLINE DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2013-12-04 EP disclosed
WO-2012101068-A1 NOVEL TETRAHYDROQUINOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2012-08-02 WO disclosed