SCHEMBL12465803

SCHEMBL12465803

CC1(C)CCOc2ccc(C(Br)C=O)cc21

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
RARA P10276 4/20 0.44
RARB P10826 4/20 0.44
RARG P13631 4/20 0.44
RXRA P19793 2/20 0.41
CYP26A1 O43174 1/20 0.39
CYP26B1 Q9NR63 1/20 0.39
AKR1B1 P15121 1/20 0.34
HNF4A P41235 1/20 0.34
PTGS1 P23219 1/20 0.33
PTGS2 P35354 1/20 0.33
SSTR5 P35346 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10555380 0.82 RARA (0.44) RARARARBRARGRXRACYP26A1
SCHEMBL12715255 0.79 RARA (0.46) RARARARBRARGRXRACYP26A1
SCHEMBL3819800 0.79 RXRA (0.49) RARARARBRARGRXRACYP26A1
SCHEMBL12465699 0.77 SSTR5 (0.33) PTGS1PTGS2SSTR5
SCHEMBL10408115 0.77 RARA (0.47) RARARARBRARGRXRACYP26A1
SCHEMBL6144459 0.76 RARA (0.41) RARARARBRARGRXRACYP26A1
SCHEMBL6144456 0.76 RARA (0.41) RARARARBRARGRXRACYP26A1
SCHEMBL6144462 0.76 RARA (0.41) RARARARBRARGRXRACYP26A1
SCHEMBL289444 0.75 RARB (0.55) RARARARBRARGRXRACYP26A1
SCHEMBL3998188 0.72 CYP26A1 (0.49) RARARARBRARGRXRACYP26A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2670744-A1 PYRROLE DERIVATIVES USED AS MODULATORS OF ALPHA7 NACHR Lupin Limited (IN) 2013-12-11 EP disclosed
WO-2012104782-A1 PYRROLE DERIVATIVES USED AS MODULATORS OF ALPHA7 NACHR LUPIN LIMITED (IN) 2012-08-09 WO disclosed