SCHEMBL1246916

SCHEMBL1246916

O=C(O)N1CCN(C(=O)c2cnc(-c3ccccc3)nc2)CC1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2B P41595 1/20 0.54
SLC6A7 Q99884 6/20 0.51
ALDH1A1 P00352 3/20 0.51
TSHR P16473 2/20 0.51
HPGD P15428 4/20 0.51
MAPK1 P28482 3/20 0.50
POLB P06746 2/20 0.50
CKS1B P61024 1/20 0.50
SKP1 P63208 1/20 0.50
SKP2 Q13309 1/20 0.50
TACR3 P29371 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
FASN P49327 2/20 0.48
PRKAB2 O43741 1/20 0.47
PRKAG1 P54619 1/20 0.47
PRKAA2 P54646 1/20 0.47
PRKAA1 Q13131 1/20 0.47
PRKAG3 Q9UGI9 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1246568 0.84 SIGMAR1 (0.66) HTR2BHPGDMAPK1
SCHEMBL4298854 0.81 HPGDS (0.59) HTR2BALDH1A1POLBCKS1BSKP1
SCHEMBL4719812 0.80 MAPK1 (0.77) SLC6A7ALDH1A1TSHRHPGDMAPK1
SCHEMBL3110048 0.79 KMT2A (0.52) HTR2BSLC6A7ALDH1A1TSHRHPGD
SCHEMBL1938606 0.79 HPGD (0.70) ALDH1A1TSHRHPGDMAPK1POLB
SCHEMBL20788243 0.74 SMN1; SMN2 (0.48) ALDH1A1HPGDPOLBL3MBTL1PRKAB2
SCHEMBL2678752 0.74 HPGD (0.75) ALDH1A1TSHRHPGDMAPK1POLB
SCHEMBL10721898 0.73 MAPK1 (0.85) SLC6A7ALDH1A1TSHRHPGDMAPK1
SCHEMBL1244776 0.73 LDHA (0.62) TSHRHPGDMEN1KMT2A
SCHEMBL252026 0.72 HPGD (0.79) ALDH1A1TSHRHPGDMAPK1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2286221-A2 METHODS FOR ASSAYING COMPOUNDS OR AGENTS FOR ABILITY TO DISPLACE POTENT LIGANDS OF HEMATOPOIETIC PROSTAGLANDIN D SYNTHASE Cayman Chemical Company (US) 2011-02-23 EP disclosed
WO-2009140364-A2 METHODS FOR ASSAYING COMPOUNDS OR AGENTS FOR ABILITY TO DISPLACE POTENT LIGANDS OF HEMATOPOIETIC PROSTAGLANDIN D SYNTHASE CAYMAN CHEMICAL COMPANY (US) 2009-11-19 WO disclosed