SCHEMBL12469894

SCHEMBL12469894

Brc1cccc(-c2nnnc(-c3ccccc3)c2-c2ccccc2)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.50
RAB9A P51151 4/20 0.50
SMN1; SMN2 Q16637 4/20 0.50
TSHR P16473 2/20 0.50
TP53 P04637 1/20 0.50
IDO1 P14902 2/20 0.49
GABRG2 P18507 4/20 0.46
GABRB3 P28472 4/20 0.46
GABRA5 P31644 4/20 0.46
GABRA3 P34903 4/20 0.46
GABRA1 P14867 1/20 0.46
MAOB P27338 1/20 0.42
LMNA P02545 4/20 0.42
HTT P42858 3/20 0.42
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
MAPT P10636 3/20 0.41
ALDH1A1 P00352 2/20 0.41
HPGD P15428 1/20 0.41
CYP1A2 P05177 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17287226 0.83 ALDH1A1 (0.54) NPC1RAB9ASMN1; SMN2TP53LMNA
SCHEMBL500715 0.82 LMNA (0.56) NPC1RAB9ASMN1; SMN2TP53LMNA
SCHEMBL22360955 0.80 LMNA (0.54) NPC1RAB9ASMN1; SMN2LMNAHTT
SCHEMBL29446652 0.79 IDO1 (0.56) NPC1RAB9ASMN1; SMN2TSHRTP53
SCHEMBL23162526 0.79 IDO1 (0.56) NPC1RAB9ASMN1; SMN2TSHRTP53
SCHEMBL26352410 0.79 NPC1 (0.53) NPC1RAB9ASMN1; SMN2TSHRTP53
Water SCHEMBL28964119 0.78 LMNA (0.52) NPC1RAB9ASMN1; SMN2LMNAHTT
Water SCHEMBL28150223 0.78 LMNA (0.52) NPC1RAB9ASMN1; SMN2LMNAHTT
SCHEMBL19497384 0.76 RAB9A (0.53) NPC1RAB9ASMN1; SMN2TSHRTP53
SCHEMBL15862445 0.74 NPC1 (0.41) NPC1RAB9ASMN1; SMN2MAOBLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2787053-B1 Polymeric materials MERCK PATENT GMBH (DE) 2018-11-21 EP disclosed
EP-2627732-B1 MATERIALS FOR ORGANIC ELECTROLUMINESCENCE DEVICES MERCK PATENT GMBH (DE) 2017-12-20 EP disclosed
CN-103228759-B Material for organic electroluminescent device 弗朗霍夫应用科学研究促进协会 2016-10-26 CN disclosed
EP-2787053-A1 Polymeric materials Merck Patent GmbH (DE) 2014-10-08 EP disclosed
US-8786181-B2 Materials for organic electroluminescent devices MERCK PATENT GMBH (DE) 2014-07-22 US disclosed
EP-2627732-A1 MATERIALS FOR ORGANIC ELECTROLUMINESCENCE DEVICES Merck Patent GmbH (DE) 2013-08-21 EP disclosed
US-20130207095-A1 MATERIALS FOR ORGANIC ELECTROLUMINESCENT DEVICES Fraunhofer-Gesellschaft Forderung E.V. (DE) 2013-08-15 US disclosed
WO-2012048900-A1 MATERIALS FOR ORGANIC ELECTROLUMINESCENCE DEVICES FRAUNHOFER-GESELLSCHAFT ZUR FÖRDERUNG DER ANGEWANDTEN FORSCHUNG E.V. . (DE) 2012-04-19 WO disclosed