SCHEMBL12470477

SCHEMBL12470477

Cc1ccc(Nc2ccc(C)cc2F)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 3/20 0.46
EGFR P00533 1/20 0.46
GAA P10253 4/20 0.46
MAPT P10636 4/20 0.46
TDP1 Q9NUW8 2/20 0.46
RAPGEF4 Q8WZA2 1/20 0.45
HPGD P15428 1/20 0.45
SOS1 Q07889 1/20 0.45
NPC1 O15118 2/20 0.44
RAB9A P51151 1/20 0.44
KDM4E B2RXH2 2/20 0.44
GFER P55789 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
MAP2K2 P36507 1/20 0.43
MAP2K1 Q02750 1/20 0.43
MAPK1 P28482 1/20 0.43
DHODH Q02127 3/20 0.43
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
AKR1C3 P42330 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18590739 0.98 SOS1 (0.46) L3MBTL1EGFRGAAMAPTTDP1
SCHEMBL13456177 0.82 SOS1 (0.73) SOS1
SCHEMBL18591949 0.82 MAPT (0.45) GAAMAPTTDP1HPGDNPC1
SCHEMBL18590729 0.79 MEN1 (0.42) EGFRGAAMAPTRAPGEF4NPC1
SCHEMBL3371377 0.79 MAPT (0.60) L3MBTL1EGFRGAAMAPTTDP1
SCHEMBL5667044 0.78 RAPGEF4 (0.63) L3MBTL1EGFRGAAMAPTTDP1
SCHEMBL30146931 0.78 RAPGEF4 (0.63) L3MBTL1EGFRGAAMAPTTDP1
SCHEMBL27786542 0.78 MAP2K2 (0.44) RAPGEF4SOS1MAP2K2MAP2K1MAPK1
SCHEMBL22563167 0.78 PGR (0.42) RAPGEF4MAP2K2MAP2K1DHODHMEN1
SCHEMBL5028501 0.77 RAPGEF4 (0.61) L3MBTL1EGFRGAAMAPTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017034023-A1 COMPLEX AND OPTICAL ELEMENT 国立大学法人京都大学 2017-03-02 WO disclosed
US-20130193382-A1 COMPOUNDS FOR ELECTRONIC DEVICES MERCK PATENT GMBH (DE) 2013-08-01 US disclosed
WO-2012048780-A1 COMPOUNDS FOR ELECTRONIC DEVICES MERCK PATENT GMBH (DE) 2012-04-19 WO disclosed