SCHEMBL12470702

SCHEMBL12470702

CC(C)(C)OC(=O)Nc1ccc2c(c1)C(O)CC(C)(C)O2

nearest known ligand 0.62

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 6/20 0.62
SIRT1 Q96EB6 3/20 0.62
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA9 Q16790 1/20 0.44
HCRTR1 O43613 1/20 0.40
HCRTR2 O43614 1/20 0.40
SLC10A2 Q12908 1/20 0.40
TRPV1 Q8NER1 1/20 0.40
RORC P51449 8/20 0.39
TLR3 O15455 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21788610 0.87 SIRT2 (0.61) SIRT2SIRT1CA12CA1CA9
SCHEMBL17781644 0.78 HPGD (0.45) SIRT2TRPV1MEN1KMT2A
SCHEMBL31371256 0.75 SIRT2 (1.00) SIRT2SIRT1TRPV1RORC
SCHEMBL11904033 0.75 MAPT (0.53) SIRT2SIRT1CA12CA1CA9
SCHEMBL6958495 0.74 SIRT2 (0.48) SIRT2SIRT1CA12CA1CA9
SCHEMBL29921932 0.73 KDM4E (0.53) SIRT2SIRT1CA12CA1CA9
SCHEMBL20809519 0.72 PYGL (0.47) SIRT2SIRT1CA12CA1CA9
SCHEMBL14484923 0.71 NPC1 (0.66) MEN1KMT2A
SCHEMBL8342099 0.71 CYP1A2 (0.63) MEN1KMT2A
SCHEMBL19859973 0.70 CA12 (0.46) SIRT2SIRT1CA12CA1CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012107262-A1 DIHYDROBENZOPYRAN, THIOCHROMAN, TETRAHYDROQUINOLEINE AND TETRAHYDRONAPHTALENE DERIVATIVES AND THEIR USE IN ANTICANCER THERAPY UNIVERSITE DE LIEGE (BE) 2012-08-16 WO disclosed