SCHEMBL19859973

SCHEMBL19859973

CC1Cc2ccc(NC(=O)OC(C)(C)C)cc2C1O

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
CA9 Q16790 1/20 0.46
NR1I3 Q14994 5/20 0.43
SLC10A2 Q12908 1/20 0.41
MMP8 P22894 6/20 0.41
MMP3 P08254 3/20 0.41
SIRT2 Q8IXJ6 2/20 0.41
SIRT1 Q96EB6 2/20 0.41
BRD4 O60885 1/20 0.40
CREBBP Q92793 1/20 0.40
HCRTR1 O43613 1/20 0.40
HCRTR2 O43614 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
CYP17A1 P05093 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27975122 0.79 MMP8 (0.47) CA12CA1CA9NR1I3MMP8
SCHEMBL14904889 0.78 NPC1 (0.47) CA12CA1CA9NR1I3SLC10A2
SCHEMBL30476642 0.77 NPC1 (0.53) CA12CA1CA9NR1I3NPC1
SCHEMBL19996133 0.77 NPC1 (0.53) CA12CA1CA9NR1I3NPC1
SCHEMBL1114945 0.76 RAB9A (0.56) CA12CA1CA9NR1I3MMP8
SCHEMBL15985239 0.75 ACHE (0.49) CA12CA1CA9NR1I3MMP8
SCHEMBL20809519 0.75 PYGL (0.47) CA12CA1CA9NR1I3SLC10A2
SCHEMBL7046627 0.74 CA12 (0.47) CA12CA1CA9NR1I3MMP8
SCHEMBL31169451 0.74 NPC1 (0.57) NR1I3NPC1RAB9A
SCHEMBL13783463 0.74 NPC1 (0.60) NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9890147-B2 2,3-benzodiazepines BAYER PHARMA AKTIENGESELLSHAFT (DE) 2018-02-13 US disclosed