SCHEMBL12470902

SCHEMBL12470902

Cc1oc2cc3c(cc2c1C(=O)Nc1ccccc1Br)OCO3

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 9/20 0.48
MAPT P10636 5/20 0.47
RAB9A P51151 8/20 0.45
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
PTGS2 P35354 1/20 0.44
KDM4E B2RXH2 4/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
NFKB1 P19838 1/20 0.42
NFKB2 Q00653 1/20 0.42
RELA Q04206 1/20 0.42
ALDH1A1 P00352 5/20 0.41
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2C9 P11712 2/20 0.41
CYP2C19 P33261 2/20 0.41
HTT P42858 2/20 0.41
LMNA P02545 3/20 0.41
HPGD P15428 1/20 0.41
TSHR P16473 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12469832 0.80 MEN1 (0.59) NPC1MAPTRAB9AMEN1KMT2A
SCHEMBL12470257 0.73 ALDH1A1 (0.44) MAPTRAB9AMEN1KMT2AKDM4E
SCHEMBL21829001 0.69 MAPT (0.70) NPC1MAPTRAB9AMEN1KMT2A
SCHEMBL21829009 0.68 MAPT (0.68) NPC1MAPTRAB9AMEN1KMT2A
SCHEMBL21829027 0.64 MAPT (1.00) NPC1MAPTRAB9AMEN1KMT2A
SCHEMBL21829017 0.64 MAPT (0.67) NPC1MAPTRAB9AMEN1KMT2A
SCHEMBL29959525 0.64 MAPT (1.00) NPC1MAPTRAB9AMEN1KMT2A
SCHEMBL21829008 0.64 MAPT (0.67) NPC1MAPTRAB9AMEN1KMT2A
SCHEMBL21828975 0.64 MAPT (0.70) NPC1MAPTRAB9AMEN1KMT2A
SCHEMBL21828973 0.64 MAPT (0.70) NPC1MAPTRAB9AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012049555-A1 SPIROCYCLIC COMPOUNDS AS VOLTAGE-GATED SODIUM CHANNEL MODULATORS LUPIN LIMITED (IN) 2012-04-19 WO disclosed