SCHEMBL12469832

SCHEMBL12469832

Cc1oc2ccccc2c1C(=O)Nc1ccccc1Br

nearest known ligand 0.59

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.59
NPC1 O15118 1/20 0.59
RAB9A P51151 1/20 0.59
KMT2A Q03164 1/20 0.59
CYP2C19 P33261 6/20 0.54
MAOB P27338 1/20 0.52
EYA3 Q99504 3/20 0.49
ALDH1A1 P00352 3/20 0.46
LMNA P02545 1/20 0.45
MAPT P10636 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
TP53 P04637 1/20 0.44
ATM Q13315 1/20 0.44
EGFR P00533 1/20 0.43
CYP2C9 P11712 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12470902 0.80 NPC1 (0.48) MEN1NPC1RAB9AKMT2ACYP2C19
SCHEMBL3263341 0.77 CYP2C19 (0.58) NPC1RAB9ACYP2C19EYA3ALDH1A1
SCHEMBL30753455 0.74 CYP2C19 (0.54) MEN1KMT2ACYP2C19MAOBEYA3
SCHEMBL30753472 0.74 CYP2C19 (0.54) MEN1NPC1RAB9AKMT2ACYP2C19
SCHEMBL1398779 0.72 CYP2C19 (0.63) MEN1RAB9AKMT2ACYP2C19EYA3
SCHEMBL9657351 0.72 CYP2C19 (0.63) MEN1NPC1RAB9AKMT2ACYP2C19
SCHEMBL18018241 0.71 CYP2C19 (0.61) MEN1KMT2ACYP2C19EYA3ALDH1A1
SCHEMBL4670295 0.71 CYP2C19 (0.61) CYP2C19EYA3ALDH1A1CYP2C9
SCHEMBL20441188 0.71 CYP2C19 (0.61) MEN1KMT2ACYP2C19EYA3LMNA
SCHEMBL1919253 0.71 CYP2C19 (0.61) MEN1KMT2ACYP2C19EYA3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012049555-A1 SPIROCYCLIC COMPOUNDS AS VOLTAGE-GATED SODIUM CHANNEL MODULATORS LUPIN LIMITED (IN) 2012-04-19 WO disclosed