SCHEMBL12474256

SCHEMBL12474256

CC(=O)O[C@@H]1OCc2cc(OS(=O)(=O)C(F)(F)F)ccc21

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.42
AKR1C3 P42330 1/20 0.37
DRD2 P14416 6/20 0.37
DRD3 P35462 6/20 0.37
HTR1D P28221 1/20 0.37
DRD4 P21917 3/20 0.36
CHRM1 P11229 2/20 0.36
CXCR2 P25025 2/20 0.35
CXCR1 P25024 1/20 0.34
DRD1 P21728 1/20 0.34
DRD5 P21918 1/20 0.34
HTR2C P28335 1/20 0.33
HTR7 P34969 1/20 0.33
HTR6 P50406 1/20 0.33
GABRA1 P14867 1/20 0.33
GABRB2 P47870 1/20 0.33
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27984641 0.76 MAPK1 (0.41) AKR1C3GABRA1GABRB2CA2
SCHEMBL3718724 0.75 HSD11B1 (0.41) HSD11B1AKR1C3DRD2DRD3DRD4
Methylamine SCHEMBL27336813 0.74 MAPK1 (0.40) AKR1C3GABRA1GABRB2
SCHEMBL1707740 0.72 HSD11B1 (0.41) HSD11B1AKR1C3DRD2DRD3HTR1D
SCHEMBL3655498 0.72 HSD11B1 (0.37) HSD11B1DRD2DRD3HTR1DDRD4
SCHEMBL3024960 0.70 RORC (0.43) HSD11B1DRD2DRD3DRD4DRD1
SCHEMBL3024958 0.70 RORC (0.43) HSD11B1DRD2DRD3DRD4DRD1
SCHEMBL31136597 0.68 HSD11B1 (0.41) HSD11B1DRD2DRD3HTR1DDRD4
SCHEMBL3533741 0.68 DRD2 (0.43) AKR1C3DRD2DRD3HTR1DDRD4
SCHEMBL3533743 0.68 DRD2 (0.43) AKR1C3DRD2DRD3HTR1DDRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2675774-A1 PRODUCTION METHOD OF OPTICALLY ACTIVE DIHYDROBENZOFURAN DERIVATIVE Takeda Pharmaceutical Company Limited (JP) 2013-12-25 EP disclosed
WO-2012111849-A1 PRODUCTION METHOD OF OPTICALLY ACTIVE DIHYDROBENZOFURAN DERIVATIVE TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-08-23 WO disclosed