SCHEMBL12484192

SCHEMBL12484192

FC(F)(F)Oc1ccc(CC2NCCc3ccsc32)cc1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.42
OPRD1 P41143 1/20 0.42
OPRK1 P41145 1/20 0.42
ALDH1A1 P00352 1/20 0.39
SLC22A1 O15245 1/20 0.37
PRCP P42785 1/20 0.37
HTR2C P28335 2/20 0.37
KDM1A O60341 2/20 0.36
DRD2 P14416 1/20 0.36
DRD4 P21917 1/20 0.36
KCNH2 Q12809 1/20 0.36
BCHE P06276 1/20 0.36
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 1/20 0.35
MAPT P10636 1/20 0.35
PKM P14618 1/20 0.35
KMT2A Q03164 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
TBXA2R P21731 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12486539 0.84 BCHE (0.45) BCHEKDM4EMEN1MAPTPKM
SCHEMBL12485441 0.80 SLC22A1 (0.43) SLC22A1PRCPKDM1ADRD2DRD4
SCHEMBL4709300 0.79 SLC22A1 (0.59) SLC22A1PRCPKDM1A
SCHEMBL12485294 0.75 SLC22A1 (0.42) SLC22A1PRCPKDM1ADRD2DRD4
SCHEMBL12485208 0.73 SLC22A1 (0.37) SLC22A1PRCPKDM1ADRD2DRD4
SCHEMBL12484520 0.73 BCHE (0.54) BCHEKDM4EMAPTPKM
SCHEMBL12486551 0.72 CHRM4 (0.53) OPRM1DRD2TBXA2R
Hydrochloric Acid SCHEMBL12484284 0.72 SLC22A1 (0.36) SLC22A1PRCPKDM1ADRD2DRD4
SCHEMBL12486444 0.72 GAA (0.37) SLC22A1PRCPKDM1ADRD2DRD4
SCHEMBL1364766 0.72 L3MBTL1 (0.43) HTR2CKDM1ATBXA2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012114252-A1 NOVEL INDOLE AND PYRROLOPYRIDINE AMIDES ACTELION PHARMACEUTICALS LTD (CH) 2012-08-30 WO disclosed