SCHEMBL12486252

SCHEMBL12486252

CCc1ccc(CC2NCCc3ccsc32)cn1

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.38
KDM4E B2RXH2 1/20 0.38
MAPT P10636 1/20 0.38
HTT P42858 1/20 0.38
SLC22A1 O15245 1/20 0.34
PRCP P42785 1/20 0.34
DRD2 P14416 3/20 0.33
DRD4 P21917 2/20 0.33
MEN1 O00255 1/20 0.33
ABL1 P00519 1/20 0.33
ALPL P05186 1/20 0.33
KMT2A Q03164 1/20 0.33
RIN1 Q13671 1/20 0.33
KDM1A O60341 1/20 0.33
BCHE P06276 1/20 0.33
TBXA2R P21731 1/20 0.32
TAAR1 Q96RJ0 2/20 0.32
HTR1A P08908 1/20 0.32
HTR7 P34969 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12486444 0.85 GAA (0.37) GAAKDM4EMAPTHTTSLC22A1
Hydrochloric Acid SCHEMBL12485366 0.84 GAA (0.36) GAAKDM4EMAPTHTTSLC22A1
SCHEMBL12486377 0.83 SLC22A1 (0.35) GAAKDM4EMAPTHTTSLC22A1
SCHEMBL12485441 0.77 SLC22A1 (0.43) GAASLC22A1PRCPDRD2DRD4
SCHEMBL4709300 0.75 SLC22A1 (0.59) SLC22A1PRCPKDM1A
SCHEMBL12486539 0.75 BCHE (0.45) KDM4EMAPTMEN1KMT2ABCHE
SCHEMBL12484520 0.72 BCHE (0.54) GAAKDM4EMAPTHTTBCHE
SCHEMBL12485208 0.72 SLC22A1 (0.37) GAASLC22A1PRCPDRD2DRD4
SCHEMBL12485294 0.72 SLC22A1 (0.42) GAASLC22A1PRCPDRD2DRD4
SCHEMBL12486244 0.72 TAAR1 (0.33) GAADRD2MEN1KMT2ATAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012114252-A1 NOVEL INDOLE AND PYRROLOPYRIDINE AMIDES ACTELION PHARMACEUTICALS LTD (CH) 2012-08-30 WO disclosed