SCHEMBL12486351

SCHEMBL12486351

CS(=O)(=O)OC/C(=C\c1ccccc1)c1ccc(F)cc1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 3/20 0.49
AKR1C3 P42330 2/20 0.43
AKR1C2 P52895 1/20 0.43
AKR1C1 Q04828 1/20 0.43
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
LMNA P02545 1/20 0.41
CYP1A2 P05177 1/20 0.41
MAPT P10636 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
MTNR1A P48039 2/20 0.40
MTNR1B P49286 2/20 0.40
POLB P06746 1/20 0.40
BRAF P15056 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12486353 1.00 PTGS2 (0.49) PTGS2AKR1C3AKR1C2AKR1C1MEN1
SCHEMBL12486822 0.74 NQO2 (0.47) PTGS2MEN1KMT2ALMNACYP1A2
SCHEMBL27516701 0.73 TSHR (0.36) PTGS2LMNANPSR1MTNR1AMTNR1B
SCHEMBL2544347 0.72 PTPN1 (0.48) MEN1KMT2ALMNAPOLB
SCHEMBL14045283 0.71 AKR1C3 (0.55) PTGS2AKR1C3AKR1C2AKR1C1
SCHEMBL1486709 0.69 MTNR1A (0.51) AKR1C1MEN1KMT2AMTNR1AMTNR1B
SCHEMBL9848407 0.67 MTNR1A (0.49) AKR1C1MEN1KMT2AMTNR1AMTNR1B
Methanesulfonic Acid Ethyl Ester SCHEMBL27549033 0.67 KMT2A (0.41) PTGS2KMT2ACYP1A2CYP2C19
SCHEMBL28483644 0.66 PTGS2 (0.44) PTGS2MEN1KMT2ALMNACYP1A2
SCHEMBL9859922 0.66 ESR1 (0.67) PTGS2MEN1KMT2AMAPTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012117421-A1 HISTONE DEACETYLASE INHIBITORS ORCHID RESEARCH LABORATORIES LTD (IN) 2012-09-07 WO disclosed