SCHEMBL12517697

SCHEMBL12517697

Cn1cc(-n2ccc(=O)c(Cc3cccc(NC(N)=O)c3)n2)cn1

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 8/20 0.38
JAK3 P52333 4/20 0.38
JAK1 P23458 2/20 0.38
GPR142 Q7Z601 1/20 0.38
MET P08581 2/20 0.37
AURKA O14965 1/20 0.36
ALK Q9UM73 1/20 0.36
DHX9 Q08211 1/20 0.36
JAK2 O60674 1/20 0.36
NTRK1 P04629 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL165695 0.92 PARP1 (0.40) PARP1JAK3JAK1GPR142MET
SCHEMBL2265122 0.91 PARP1 (0.38) PARP1JAK3JAK1GPR142MET
SCHEMBL2365347 0.90 PARP1 (0.47) PARP1JAK3MET
SCHEMBL13465733 0.90 MET (0.40) PARP1JAK3JAK1MET
SCHEMBL13274893 0.89 HTR1A (0.44) PARP1MET
SCHEMBL2361582 0.89 PARP1 (0.49) PARP1JAK3JAK2
SCHEMBL2271983 0.89 PARP1 (0.41) PARP1JAK3JAK1METAURKA
SCHEMBL13465435 0.88 PARP1 (0.49) PARP1JAK3JAK1METJAK2
SCHEMBL255442 0.87 RORC (0.40) PARP1AURKA
SCHEMBL2269942 0.87 SMN1; SMN2 (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011084402-A1 TYROSINE KINASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2011-07-14 WO disclosed