SCHEMBL12527177

SCHEMBL12527177

Fc1ccccc1-c1cc(-c2cncc(-c3cnn(C4CCNCC4)c3)c2)c2nccnc2n1

nearest known ligand 0.58

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAP4K1 Q92918 3/20 0.58
ALK Q9UM73 3/20 0.46
MET P08581 3/20 0.46
CHRNB2 P17787 3/20 0.46
CHRNA4 P43681 3/20 0.46
PAK1 Q13153 2/20 0.45
MAP4K3 Q8IVH8 1/20 0.45
JAK2 O60674 1/20 0.45
ABL1 P00519 1/20 0.45
JAK1 P23458 1/20 0.45
TYK2 P29597 1/20 0.45
JAK3 P52333 1/20 0.45
PAK4 O96013 1/20 0.44
IRAK4 Q9NWZ3 1/20 0.43
GRK2 P25098 1/20 0.43
GRK5 P34947 1/20 0.43
KCNH2 Q12809 2/20 0.43
PIM1 P11309 1/20 0.43
INPPL1 O15357 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2320474 0.89 MAP4K1 (0.53) MAP4K1ALKMETCHRNB2CHRNA4
SCHEMBL12524281 0.89 MAP4K1 (0.47) MAP4K1MET
Hydrochloric Acid SCHEMBL13834975 0.88 MAP4K1 (0.52) MAP4K1ALKMETCHRNB2CHRNA4
SCHEMBL320855 0.83 MAP4K1 (0.56) MAP4K1ALKMETCHRNB2CHRNA4
SCHEMBL12495538 0.83 MAP4K1 (0.49) MAP4K1METJAK2JAK3
SCHEMBL12495426 0.82 MAP4K1 (0.51) MAP4K1ALKMETPIM1
SCHEMBL2321067 0.80 INPPL1 (0.50) MAP4K1ALKMETCHRNB2CHRNA4
SCHEMBL2324841 0.80 MAP4K3 (0.47) MAP4K1ALKMETCHRNB2CHRNA4
Hydrochloric Acid SCHEMBL2324061 0.80 INPPL1 (0.49) MAP4K1ALKMETCHRNB2CHRNA4
SCHEMBL12524282 0.79 MET (0.49) MAP4K1METINPPL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012119690-A1 PYRIDO [2, 3 - B] PYRAZINE DERIVATIVES AND THEIR THERAPEUTICAL USES MERCK PATENT GMBH (DE) 2012-09-13 WO disclosed