SCHEMBL1256199

SCHEMBL1256199

Cn1nnc2ccc(C(=O)O)cc21

nearest known ligand 0.76

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HCAR3 P49019 13/20 0.76
HPGD P15428 4/20 0.53
HCAR2 Q8TDS4 1/20 0.53
MEN1 O00255 1/20 0.50
RAB9A P51151 1/20 0.50
KMT2A Q03164 1/20 0.50
POLB P06746 1/20 0.49
MAPT P10636 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL599138 0.86 HCAR3 (1.00) HCAR3HPGDHCAR2MEN1RAB9A
SCHEMBL12349868 0.86 HCAR3 (0.57) HCAR3HPGDMEN1RAB9AKMT2A
SCHEMBL29751355 0.85 HCAR3 (0.55) HCAR3HPGDMEN1RAB9AKMT2A
SCHEMBL2884485 0.82 HCAR3 (0.53) HCAR3HPGDMEN1RAB9AKMT2A
SCHEMBL2852713 0.81 HSD17B10 (0.56) HCAR3HPGDHCAR2POLB
SCHEMBL6184550 0.80 HCAR3 (0.80) HCAR3HPGDHCAR2
SCHEMBL8712864 0.80 NPC1 (0.55) HCAR3HPGDMEN1RAB9AKMT2A
SCHEMBL7232454 0.79 HCAR3 (0.53) HCAR3HPGDHCAR2KMT2A
SCHEMBL6182902 0.79 HCAR3 (0.78) HCAR3HPGDHCAR2MEN1RAB9A
SCHEMBL11391092 0.79 HCAR3 (0.53) HCAR3HPGDHCAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 37 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4704830-A2 MRGPRX2 INHIBITORS AND METHODS OF USE THEREOF Septerna, Inc. (US) 2026-03-11 EP disclosed
WO-2024226914-A2 MRGPRX2 ANTAGONISTS AND METHODS OF USE THEREOF SEPTERNA, INC. (US) 2024-10-31 WO disclosed
CN-117858877-A C-linked inhibitors of ENL/AF9 YEATS 桥梁药品有限公司 2024-04-09 CN disclosed
EP-4271672-A1 CARBOXY-BENZIMIDAZOLE GLP-1R MODULATING COMPOUNDS GILEAD SCIENCES, INC. (US) 2023-11-08 EP disclosed
US-20230322722-A1 MODULATORS OF MYC FAMILY PROTO-ONCOGENE PROTEIN NALO THERAPEUTICS (US) 2023-10-12 US disclosed
US-20230322722-A1 MODULATORS OF MYC FAMILY PROTO-ONCOGENE PROTEIN NALO THERAPEUTICS (US) 2023-10-12 US disclosed
EP-4204411-A1 MODULATORS OF MYC FAMILY PROTO-ONCOGENE PROTEIN Nalo Therapeutics (US) 2023-07-05 EP disclosed
WO-2022225941-A1 CARBOXY-BENZIMIDAZOLE GLP-1R MODULATING COMPOUNDS GILEAD SCIENCES, INC. (US) 2022-10-27 WO disclosed
WO-2022046861-A1 MODULATORS OF MYC FAMILY PROTO-ONCOGENE PROTEIN NALO THERAPEUTICS (US) 2022-03-03 WO disclosed
EP-3002283-B1 THIAZOLE DERIVATIVES KYOWA HAKKO KIRIN CO LTD (JP) 2017-06-14 EP disclosed
CN-1681805-A Novel imidazole compounds as transforming growth factor (TGF) inhibitors PFIZER PROD INC (US) 2005-10-12 CN disclosed
EP-1542990-A1 NOVEL IMIDAZOLE COMPOUNDS AS TRANSFORMING GROWTH FACTOR (TGF) INHIBITORS Pfizer Products Inc. (US) 2005-06-22 EP disclosed
WO-2004111046-A2 THIAZOLES AS INHIBITORS OF THE ALK- 5 RECEPTOR SMITHKLINE BEECHAM CORPORATION (US) 2004-12-23 WO disclosed
US-20040106608-A1 Novel imidazole compounds as transforming growth factor (TGF) inhibitors PFIZER INC 2004-06-03 US disclosed
WO-2004026859-A1 NOVEL IMIDAZOLE COMPOUNDS AS TRANSFORMING GROWTH FACTOR (TGF) INHIBITORS PFIZER PRODUCTS INC. (US) 2004-04-01 WO disclosed
EP-0408509-B1 Substituted benzonitriles CIBA GEIGY AG (CH) 1996-03-06 EP disclosed
WO-1992022536-A1 VINYLIMIDAZOLES, VINYLTRIAZOLES AND VINYLTETRAZOLES WITH A BICYCLIC SUBSTITUENT GROUP SCHERING AKTIENGESELLSCHAFT, BERLIN UND BERGKAMEN (DE) 1992-12-23 WO disclosed
EP-0518457-A1 Bicyclic substituted vinylimidazoles, -triazoles and -tetrazoles SCHERING AKTIENGESELLSCHAFT (DE) 1992-12-16 EP disclosed
US-5073574-A TETRAZOLYL SUBSTITUTED BENZONITRILES AND ANTI-TUMOR USE THEREOF CIBA-GEIGY CORPORATION (US) 1991-12-17 US disclosed
EP-0408509-A2 Substituted benzonitriles CIBA-GEIGY AG (CH) 1991-01-16 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230322722-A1 MODULATORS OF MYC FAMILY PROTO-ONCOGENE PROTEIN MYC, MYCBP, MYCBP2 HCAR3 4732/4885HPGD 3097/4885HCAR2 4842/4885
US-20040106608-A1 Novel imidazole compounds as transforming growth factor (TGF) inhibitors SMAD3, TGFBR1, TGFBR2 HCAR3 2875/4885HPGD 973/4885HCAR2 2363/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.