SCHEMBL1256644

SCHEMBL1256644

CS(=O)(=O)c1ccc(Cl)nc1

nearest known ligand 0.59

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.59
MAPT P10636 1/20 0.58
POLB P06746 1/20 0.51
ALDH1A1 P00352 8/20 0.49
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
CYP2D6 P10635 1/20 0.49
TDP1 Q9NUW8 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
GAA P10253 2/20 0.46
PKM P14618 2/20 0.46
CYP2C19 P33261 1/20 0.44
LMNA P02545 1/20 0.43
MAPK1 P28482 1/20 0.43
BLM P54132 1/20 0.43
EGFR P00533 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29977958 1.00 SMN1; SMN2 (0.59) SMN1; SMN2MAPTPOLBALDH1A1MEN1
SCHEMBL3086532 0.83 SMN1; SMN2 (0.56) SMN1; SMN2MAPTPOLBALDH1A1MEN1
SCHEMBL23845463 0.80 SMN1; SMN2 (0.53) SMN1; SMN2MAPTPOLBALDH1A1MEN1
SCHEMBL17509 0.80 SMN1; SMN2 (0.56) SMN1; SMN2MAPTPOLBALDH1A1MEN1
SCHEMBL29483829 0.80 SMN1; SMN2 (0.56) SMN1; SMN2MAPTPOLBALDH1A1MEN1
SCHEMBL14744375 0.79 MAPT (0.64) SMN1; SMN2MAPTPOLBALDH1A1MEN1
SCHEMBL7808800 0.79 NAPRT (0.51) SMN1; SMN2MAPTALDH1A1BLMEGFR
SCHEMBL2633979 0.78 KDM4E (0.59) SMN1; SMN2MAPTPOLBALDH1A1MEN1
SCHEMBL4804914 0.78 SMN1; SMN2 (0.59) SMN1; SMN2MAPTPOLBALDH1A1MEN1
Hydrochloric Acid SCHEMBL4803286 0.78 SMN1; SMN2 (0.55) SMN1; SMN2MAPTPOLBALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 121 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117903115-A Sulfone-substituted heterocyclic structure compound, preparation method thereof and application thereof in medicine 上海致根医药科技有限公司 2024-04-19 CN disclosed
EP-3419972-B1 GLYCOSIDASE INHIBITORS ASCENEURON SA (CH) 2023-07-26 EP disclosed
US-11612599-B2 Glycosidase inhibitors ASCENEURON SA (CH) 2023-03-28 US disclosed
CN-110494431-B Azacyclo derivative, preparation method and medical application thereof 苏州浦合医药科技有限公司 2022-11-04 CN disclosed
EP-3419971-B1 GLYCOSIDASE INHIBITORS ASCENEURON SA (CH) 2022-04-20 EP disclosed
US-11213525-B2 Linear glycosidase inhibitors ASCENEURON SA (CH) 2022-01-04 US disclosed
US-11213525-B2 Linear glycosidase inhibitors ASCENEURON SA (CH) 2022-01-04 US disclosed
US-20210186958-A1 GLYCOSIDASE INHIBITORS ASCENEURON SA (CH) 2021-06-24 US disclosed
US-20210077488-A1 LINEAR GLYCOSIDASE INHIBITORS ASCENEURON SA (CH) 2021-03-18 US disclosed
US-20210077488-A1 LINEAR GLYCOSIDASE INHIBITORS ASCENEURON SA (CH) 2021-03-18 US disclosed
US-20070060623-A1 antiulcer agents; proton pump inhibitors; side effect reduction; 1-[4-fluoro-5-phenyl-1-(pyridin-3-ylsulfonyl)-1H-pyrrol-3-yl]-N-methylmethanamine; superior acid secretion inhibitory effect; peptic ulcer, Zollinger-Ellison syndrome, reflux esophagitis, or symptomatic gastroesophageal reflux disease TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-03-15 US disclosed
US-20070060623-A1 antiulcer agents; proton pump inhibitors; side effect reduction; 1-[4-fluoro-5-phenyl-1-(pyridin-3-ylsulfonyl)-1H-pyrrol-3-yl]-N-methylmethanamine; superior acid secretion inhibitory effect; peptic ulcer, Zollinger-Ellison syndrome, reflux esophagitis, or symptomatic gastroesophageal reflux disease TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-03-15 US disclosed
WO-2007026916-A1 1-HETEROCYCLYLSULFONYL, 2-AMINOMETHYL, 5- (HETERO-) ARYL SUBSTITUTED 1-H-PYRROLE DERIVATIVES AS ACID SECRETION INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-03-08 WO disclosed
CN-1902196-A Thiazole derivatives KYOWA HAKKO KOGYO KK (JP) 2007-01-24 CN disclosed
EP-1700856-A1 THIAZOLE DERIVATIVE KYOWA HAKKO KOGYO CO., LTD. (JP) 2006-09-13 EP disclosed
US-20040180925-A1 Dipeptidylpeptidase-IV inhibitor KYOWA HAKKO KOGYO CO., LTD. (JP) 2004-09-16 US disclosed
EP-1354882-A1 DIPEPTIDYL PEPTIDASE IV INHIBITOR KYOWA HAKKO KOGYO CO., LTD. (JP) 2003-10-22 EP disclosed
US-6448205-B1 FOR THE DESICCATION AND/OR DEFOLIATION OF PLANTS BASF AKTIENGESELLSCHAFT (DE) 2002-09-10 US disclosed
EP-0920415-A1 SUBSTITUTED 2-PHENYLPYRIDINE AS HERBICIDE BASF AKTIENGESELLSCHAFT (DE) 1999-06-09 EP disclosed
WO-1998007700-A1 SUBSTITUTED 2-PHENYLPYRIDINE AS HERBICIDE BASF AKTIENGESELLSCHAFT (DE) 1998-02-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11213525-B2 Linear glycosidase inhibitors ENGASE, GAA, GLA SMN1; SMN2 1002/4885MAPT 38/4885POLB 2024/4885
US-11612599-B2 Glycosidase inhibitors ENGASE, GAA, GLA SMN1; SMN2 1307/4885MAPT 24/4885POLB 2755/4885
US-20210186958-A1 GLYCOSIDASE INHIBITORS ENGASE, GAA, GLA SMN1; SMN2 1307/4885MAPT 24/4885POLB 2755/4885
US-20070060623-A1 antiulcer agents; proton pump inhibitors; side effect reduction; 1-[4-fluoro-5-phenyl-1-(pyridin-3-ylsulfonyl)-1H-pyrrol-3-yl]-N-methylmethanamine; superior acid secretion inhibitory effect; peptic ulcer, Zollinger-Ellison syndrome, reflux esophagitis, or symptomatic gastroesophageal reflux disease HRH2, GIPR, HRH4 SMN1; SMN2 2144/4885MAPT 4809/4885POLB 4811/4885
US-20210077488-A1 LINEAR GLYCOSIDASE INHIBITORS ENGASE, GAA, GLA SMN1; SMN2 1002/4885MAPT 38/4885POLB 2024/4885
US-20040180925-A1 Dipeptidylpeptidase-IV inhibitor DPP4, DPP3, DPP9 SMN1; SMN2 3810/4885MAPT 3376/4885POLB 2660/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.