SCHEMBL12593274

SCHEMBL12593274

CCCCC1(CCCC)NC(=N)N(CCCNC(=O)CC2=CC=CCC2)C1=O

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
HPGD P15428 1/20 0.31
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7520071 0.80 ALDH1A1 (0.48) HPGD
SCHEMBL17551661 0.78 CNR1 (0.35)
SCHEMBL7525486 0.77 RAB9A (0.40) CYP1A2CYP2C9CYP2C19
SCHEMBL7524859 0.77 EPHX1 (0.40) CYP1A2CYP2C9CYP2C19
SCHEMBL7519666 0.77 HSD17B10 (0.36) CYP1A2CYP2C9CYP2C19MAPT
SCHEMBL7533775 0.76 ALDH1A1 (0.39) CYP1A2CYP2C9CYP2C19HPGD
SCHEMBL7524740 0.76 TYMP (0.37) CYP1A2CYP2C9CYP2C19
SCHEMBL7537395 0.75 HPGD (0.40) CYP1A2CYP2C9CYP2C19HPGD
SCHEMBL7518579 0.74 CASP2 (0.43) HPGD
SCHEMBL7522160 0.74 HPGD (0.56) HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2335701-A1 Heterocyclic aspartyl protease inhibitors Schering Corporation (US) 2011-06-22 EP disclosed