Pyridine

Pyridine

SCHEMBL126094

Cc1ccc(O)cc1S(=O)(=O)O.c1ccncc1

nearest known ligand 0.49

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 3/20 0.49
POLB P06746 2/20 0.49
RECQL P46063 1/20 0.49
LMNA P02545 1/20 0.43
HPGD P15428 1/20 0.43
HIF1A Q16665 1/20 0.43
HSD17B10 Q99714 1/20 0.43
GAA P10253 3/20 0.42
ALDH1A1 P00352 3/20 0.42
PKM P14618 1/20 0.42
GFER P55789 1/20 0.39
TSHR P16473 2/20 0.38
CYTH2 Q99418 1/20 0.37
KMT2A Q03164 2/20 0.37
MEN1 O00255 1/20 0.37
ESR1 P03372 1/20 0.37
ATM Q13315 1/20 0.37
NAPRT Q6XQN6 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.35
HTT P42858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL121153 0.86 LMNA (0.53) ESR2POLBRECQLLMNAHPGD
Water SCHEMBL3002925 0.84 LMNA (0.51) ESR2POLBRECQLLMNAHPGD
Hydrochloric Acid SCHEMBL5858440 0.84 LMNA (0.51) ESR2POLBRECQLLMNAHPGD
Ammonia Solution, Strong SCHEMBL1924833 0.84 LMNA (0.51) ESR2POLBRECQLLMNAHPGD
Dobesilic Acid SCHEMBL11655230 0.83 LMNA (0.57) POLBLMNAHPGDHIF1AHSD17B10
Acetic Acid SCHEMBL1232489 0.83 LMNA (0.47) ESR2POLBRECQLLMNAHPGD
SCHEMBL8429962 0.82 CHRM5 (0.46) ESR2POLBRECQLLMNAHPGD
Ethylene Glycol SCHEMBL6331832 0.80 LMNA (0.51) ESR2POLBRECQLLMNAHPGD
Pyridine SCHEMBL251401 0.80 TDP1 (0.47) ESR2POLBRECQLLMNAGAA
Isopropylamine SCHEMBL2350745 0.78 LMNA (0.46) ESR2POLBRECQLLMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 380 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3883913-B1 PROCESS FOR MAKING ETHERS VIA ENOL ETHERS BP PLC (GB) 2023-11-01 EP claimed
EP-3649135-B1 SYNTHESIS OF HALICHONDRINS HARVARD COLLEGE (US) 2022-12-28 EP claimed
EP-3452038-B1 PROCESS FOR THE PREPARATION OF INTERMEDIATES USEFUL IN THE PREPARATION OF HEPATITIS C VIRUS (HCV) INHIBITORS LAURUS LABS LTD (IN) 2022-07-06 EP claimed
EP-3081560-B1 TAXANES COMPOUNDS, PREPARATION METHOD THEREFOR, AND USES THEREOF JIANGSU TASLY DIYI PHARMACEUTICAL CO LTD (CN) 2021-03-24 EP claimed
EP-3421447-B1 FATTY ACID COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF SHANGHAI INST MATERIA MEDICA CAS (CN) 2021-03-24 EP claimed
EP-3072896-B1 TAXANE COMPOUND, AND PREPARATION METHOD AND USE THEREOF JIANGSU TASLY DIYI PHARMACEUTICAL CO LTD (CN) 2021-01-06 EP claimed
EP-3406586-B1 MANUFACTURING METHOD FOR HIGH-PURITY CYCLOHEXENONE LONG-CHAIN ALCOHOL TAIHO PHARMACEUTICAL CO LTD (JP) 2020-12-30 EP claimed
EP-2968294-B1 7-BENZYL-10-(2-METHYLBENZYL)-2,6,7,8,9,10-HEXAHYDROIMIDAZO[1,2-A]PYRIDO[4,3-D]PYRIMIDIN-5(3H)-ON FOR USE IN THE TREATMENT OF CANCER ONCOCEUTICS INC (US) 2019-05-01 EP claimed
EP-2714652-B1 CHIRAL SYNTHESIS OF N-{3,4-DIFLUORO-2-[(2-FLUORO-4-IODOPHENYL)AMINO]-6-METHOXYPHENYL}-1-[2,3-DIHYDROXY-PROPYL]CYCLOPROPANESULFONAMIDES BAYER IP GMBH (DE) 2018-07-18 EP claimed
EP-2883878-B1 Sulfur-containing organosilicon compound, making method, rubber compounding ingredient, and rubber composition SHINETSU CHEMICAL CO (JP) 2017-08-30 EP claimed
EP-0633878-B1 NOVEL VITAMIN D ANALOGUES LEO PHARM PROD LTD (DK) 1997-01-29 EP claimed
EP-0399818-B1 Diarylstyrylquinoline diacids MERCK FROSST CANADA INC (CA) 1995-08-16 EP claimed
EP-0348910-B1 19-substituted progesterone derivatives useful as 19-hydroxylase inhibitors MERRELL DOW PHARMA (US) 1995-05-17 EP claimed
EP-0160842-B1 2-Substituted ergoline derivatives, processes for their preparation, and their use as medicaments SCHERING AG (DE) 1994-06-22 EP claimed
EP-0379191-B1 1,3-Dioxolane benzoic acids and derivatives thereof SEARLE & CO (US) 1994-01-19 EP claimed
EP-0381989-B1 NEW 4'-EPI-4'-AMINO ANTHRACYCLINES FARMITALIA CARLO ERBA S.r.l. (IT) 1992-02-05 EP claimed
EP-0225823-B1 PROCESS FOR THE PREPARATION OF PTERIDINE DERIVATIVES RHONE-POULENC SANTE (FR) 1990-01-31 EP claimed
EP-0073061-B1 OPTICALLY UNIFORM BETA-LACTAMS, THEIR PREPARATION AND USE IN THE PREPARATION OF ANTIMICROBIAL BETA-LACTAMS, AND STARTING COMPOUNDS FOR USE IN THEIR PREPARATION F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1987-03-04 EP claimed
EP-0160842-A2 2-Substituted ergoline derivatives, processes for their preparation, and their use as medicaments SCHERING AKTIENGESELLSCHAFT (DE) 1985-11-13 EP claimed
EP-0033536-B1 6(R)-(2-(8'-ETHERIFIED-HYDROXY-2',6'-DIMETHYLPOLYHYDRO-NAPHTHYL-1')-ETHYL)-4(R)-HYDROXY-3,4,5,6-TETRAHYDRO-2H-PYRAN-2-ONES, THE HYDROXY ACID FORM OF SAID PYRANONES, THE SALTS OF SAID ACID FORM, PROCESS FOR PREPARING THE SAME AND AN ANTIHYPERCHOLESTEROLEMIC PHARMACEUTICAL COMPOSITION CONTAINING THE SAME MERCK & CO. INC. (US) 1984-09-12 EP claimed