SCHEMBL12620

SCHEMBL12620

CCOC(=O)c1nn(-c2ccccc2)c(Br)c1CS

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.57
KDM4E B2RXH2 4/20 0.57
HSD17B10 Q99714 2/20 0.57
HPGD P15428 2/20 0.57
ALOX12 P18054 2/20 0.54
TP53 P04637 1/20 0.54
CYP3A4 P08684 1/20 0.53
CYP2C9 P11712 1/20 0.53
CYP2C19 P33261 1/20 0.53
PDE4D Q08499 2/20 0.51
HTT P42858 1/20 0.50
NPC1 O15118 1/20 0.50
RAB9A P51151 1/20 0.50
MAPT P10636 2/20 0.49
ADORA1 P30542 2/20 0.49
APP P05067 1/20 0.49
ADORA2A P29274 1/20 0.49
ALOX15 P16050 1/20 0.48
CASP1 P29466 1/20 0.48
PDE4A P27815 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7732 0.89 ALDH1A1 (0.58) ALDH1A1KDM4EHSD17B10HPGDALOX12
SCHEMBL11144 0.89 ALDH1A1 (0.58) ALDH1A1KDM4EHSD17B10HPGDALOX12
SCHEMBL7613 0.80 ALDH1A1 (0.57) ALDH1A1KDM4EHSD17B10HPGDALOX12
SCHEMBL12276674 0.77 ALDH1A1 (0.46) ALDH1A1KDM4EHSD17B10HPGDALOX12
SCHEMBL13741611 0.75 KDM4E (0.64) ALDH1A1KDM4EHSD17B10HPGDALOX12
SCHEMBL4038334 0.74 ALDH1A1 (0.74) ALDH1A1KDM4EHSD17B10HPGDALOX12
SCHEMBL3262118 0.73 LMNA (0.61) ALDH1A1KDM4EHSD17B10HPGDALOX12
SCHEMBL17259302 0.73 ALDH1A1 (0.55) ALDH1A1KDM4EHSD17B10HPGDALOX12
SCHEMBL13858612 0.73 ALDH1A1 (0.61) ALDH1A1KDM4EHSD17B10HPGDALOX12
SCHEMBL11391965 0.73 MAPK1 (0.70) ALDH1A1KDM4EHSD17B10HPGDALOX12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011058149-A1 TRICYCLIC PYRAZOL AMINE DERIVATIVES MERCK SERONO S.A. (CH) 2011-05-19 WO disclosed