SCHEMBL12631365

SCHEMBL12631365

O=C(NC1COC1)C1CCN(C(=O)[C@@H]2CC[C@H](c3ccccc3)N(S(=O)(=O)c3ccccc3)C2)CC1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 2/20 0.47
HTT P42858 1/20 0.45
ALDH1A1 P00352 3/20 0.44
RAB9A P51151 2/20 0.44
KMT2A Q03164 2/20 0.44
GAA P10253 2/20 0.43
LMNA P02545 2/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
NPC1 O15118 2/20 0.42
MAPT P10636 1/20 0.39
TSHR P16473 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
MEN1 O00255 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2052027 1.00 EPHX2 (0.47) EPHX2HTTALDH1A1RAB9AKMT2A
SCHEMBL12628299 0.91 ALDH1A1 (0.52) EPHX2HTTALDH1A1RAB9AKMT2A
SCHEMBL2016241 0.91 ALDH1A1 (0.52) EPHX2HTTALDH1A1RAB9AKMT2A
SCHEMBL12631617 0.84 ALDH1A1 (0.49) EPHX2HTTALDH1A1RAB9AKMT2A
SCHEMBL12631356 0.83 HTT (0.62) HTTALDH1A1RAB9AKMT2AGAA
SCHEMBL12632349 0.83 NPC1 (0.58) HTTALDH1A1RAB9AKMT2ALMNA
SCHEMBL2013818 0.82 ALDH1A1 (0.47) EPHX2HTTALDH1A1RAB9AKMT2A
SCHEMBL12631691 0.82 ALDH1A1 (0.47) EPHX2HTTALDH1A1RAB9AKMT2A
SCHEMBL2052886 0.82 NPC1 (0.49) HTTALDH1A1RAB9AKMT2ALMNA
SCHEMBL12631377 0.82 NPC1 (0.49) HTTALDH1A1RAB9AKMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011073277-A1 PIPERIDINE ARYL SULFONAMIDE DERIVATIVES AS Kv1.3 MODULATORS EVOTEC AG (DE) 2011-06-23 WO disclosed