SCHEMBL12643148

SCHEMBL12643148

COCCn1cc(C=O)c2c(C(=O)N3CCCCC3)cccc21

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.51
HSD17B10 Q99714 8/20 0.47
ALDH1A1 P00352 7/20 0.47
KDM4E B2RXH2 7/20 0.47
GAA P10253 7/20 0.47
GLA P06280 6/20 0.47
HPGD P15428 6/20 0.47
KMT2A Q03164 4/20 0.45
MEN1 O00255 2/20 0.45
TSHR P16473 2/20 0.45
P2RX7 Q99572 5/20 0.45
IL1B P01584 4/20 0.45
SMN1; SMN2 Q16637 1/20 0.43
PKM P14618 1/20 0.42
POLB P06746 1/20 0.42
MAPT P10636 1/20 0.42
CNR2 P34972 2/20 0.41
CNR1 P21554 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12643136 0.99 NPSR1 (0.49) NPSR1HSD17B10ALDH1A1KDM4EGAA
SCHEMBL2039992 0.90 HTT (0.48) NPSR1HSD17B10ALDH1A1KDM4EGAA
SCHEMBL2041723 0.85 NPSR1 (0.56) NPSR1HSD17B10ALDH1A1KDM4EGAA
SCHEMBL2038550 0.84 NPSR1 (0.54) NPSR1HSD17B10ALDH1A1KDM4EGAA
SCHEMBL12697362 0.84 NPSR1 (0.54) NPSR1HSD17B10ALDH1A1KDM4EGAA
SCHEMBL2039777 0.81 NPSR1 (0.52) NPSR1HSD17B10ALDH1A1KDM4EGAA
SCHEMBL12643149 0.80 CNR2 (0.44) P2RX7IL1BPOLBCNR2CNR1
SCHEMBL2034386 0.76 CNR1 (0.47) ALDH1A1P2RX7IL1BMAPTCNR2
SCHEMBL12642978 0.75 POLB (0.48) ALDH1A1HPGDP2RX7IL1BSMN1; SMN2
SCHEMBL2034023 0.75 NPSR1 (0.57) NPSR1HSD17B10ALDH1A1KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011079102-A1 INDOLYL-PIPERIDINYL BENZYLAMINES AS BETA-TRYPTASE INHIBITORS SANOFI (FR) 2011-06-30 WO disclosed