SCHEMBL12653151

SCHEMBL12653151

COc1ccc(/C=C/c2ncc(NC[C@@H]3CCCN3)c(Oc3ccc(OC)cc3)n2)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C19 P33261 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HIF1A Q16665 1/20 0.38
PHLPP2 Q6ZVD8 1/20 0.38
MERTK Q12866 1/20 0.38
AKT1 P31749 1/20 0.38
EHMT2 Q96KQ7 1/20 0.35
MAPT P10636 1/20 0.34
LTA4H P09960 1/20 0.34
CHRNA3 P32297 4/20 0.34
CHRNB4 P30926 2/20 0.34
IDO1 P14902 2/20 0.34
TDO2 P48775 2/20 0.34
EGFR P00533 1/20 0.34
PDGFRB P09619 1/20 0.34
PDGFRA P16234 1/20 0.34
MAPK3 P27361 1/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1806946 1.00 CYP1A2 (0.38) CYP1A2CYP2D6CYP2C19SMN1; SMN2HIF1A
SCHEMBL1808792 0.84 CYP1A2 (0.39) CYP1A2CYP2D6CYP2C19SMN1; SMN2HIF1A
SCHEMBL12620407 0.82 DAPK1 (0.46) MERTKEGFRMAPK3MAPK1SYK
SCHEMBL12653247 0.80 ALDH1A1 (0.46) CYP1A2CYP2D6CYP2C19SMN1; SMN2HIF1A
SCHEMBL12620446 0.79 MERTK (0.36) CYP1A2CYP2D6CYP2C19SMN1; SMN2HIF1A
SCHEMBL1808671 0.79 MERTK (0.36) CYP1A2CYP2D6CYP2C19SMN1; SMN2HIF1A
SCHEMBL16519796 0.79 MERTK (0.36) CYP1A2CYP2D6CYP2C19SMN1; SMN2HIF1A
SCHEMBL1803527 0.77 LTA4H (0.41) CYP1A2CYP2D6CYP2C19SMN1; SMN2HIF1A
SCHEMBL1866415 0.77 CYP1A2 (0.37) CYP1A2CYP2D6CYP2C19SMN1; SMN2HIF1A
SCHEMBL12620422 0.76 HTR2C (0.40) CYP1A2CYP2D6CYP2C19SMN1; SMN2HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2493863-B1 PHENOXY-SUBSTITUTED PYRIMIDINES AS OPIOID RECEPTOR MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2015-02-25 EP disclosed
WO-2011053701-A1 PHENOXY-SUBSTITUTED PYRIMIDINES AS OPIOID RECEPTOR MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2011-05-05 WO disclosed