SCHEMBL12656137

SCHEMBL12656137

CCC(=O)c1cc(Cl)ncc1F

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.40
ASPH Q12797 1/20 0.40
KDM8 Q8N371 1/20 0.40
TSHR P16473 1/20 0.37
HSP90AB1 P08238 1/20 0.36
KCNQ3 O43525 6/20 0.36
KCNQ2 O43526 6/20 0.36
KCNH2 Q12809 1/20 0.35
JMJD6 Q6NYC1 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HMGCR P04035 1/20 0.34
KCNE1 P15382 4/20 0.34
KCNQ1 P51787 4/20 0.34
RXFP1 Q9HBX9 1/20 0.34
MELK Q14680 1/20 0.33
MAPT P10636 1/20 0.33
RAB9A P51151 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6223874 0.83 KDM4E (0.40) KDM4EASPHKDM8KCNQ3KCNQ2
SCHEMBL30770791 0.81 HSP90AB1 (0.37) KDM4ETSHRHSP90AB1KCNQ3KCNQ2
SCHEMBL27334085 0.81 HSP90AB1 (0.37) KDM4ETSHRHSP90AB1KCNQ3KCNQ2
SCHEMBL1809928 0.80 KDM4E (0.43) KDM4EASPHKDM8KCNQ3KCNQ2
SCHEMBL28824877 0.80 KDM4E (0.46) KDM4EASPHKDM8KCNQ3KCNQ2
SCHEMBL16712886 0.79 GABRP (0.37) KDM4EHSP90AB1ALDH1A1HMGCRMAPT
SCHEMBL21530434 0.79 JMJD6 (0.56) KDM4ETSHRJMJD6ALDH1A1MAPT
SCHEMBL20073627 0.79 NNMT (0.40) KDM4ETSHRHSP90AB1ALDH1A1HMGCR
SCHEMBL29947373 0.79 NNMT (0.40) KDM4ETSHRHSP90AB1ALDH1A1HMGCR
SCHEMBL29813883 0.78 ASPH (0.63) KDM4EASPHKDM8TSHRKCNQ3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011056725-A1 PYRIDINE DERIVATIVES AND METHODS OF USE THEREOF CRYSTALGENOMICS, INC. (KR) 2011-05-12 WO disclosed