SCHEMBL12658802

SCHEMBL12658802

COc1ccc(-c2ccc(-c3ccc(C4CCC(C)CC4)cc3)cc2F)cc1F

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TDP2 O95551 1/20 0.45
KDM1A O60341 2/20 0.42
CYP17A1 P05093 1/20 0.41
PTGS2 P35354 5/20 0.40
NAAA Q02083 4/20 0.40
PTGS1 P23219 3/20 0.40
ESR2 Q92731 1/20 0.39
FAAH O00519 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
APP P05067 1/20 0.38
PDGFRB P09619 1/20 0.38
PDGFRA P16234 1/20 0.38
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
PAX8 Q06710 1/20 0.38
PIK3CA P42336 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL802726 0.90 PTGS2 (0.43) TDP2KDM1APTGS2NAAAPTGS1
SCHEMBL10030943 0.90 PTGS2 (0.43) TDP2KDM1APTGS2NAAAPTGS1
SCHEMBL17210770 0.86 CTSK (0.39) TDP2NAAAESR2CYP3A4CYP2C9
SCHEMBL13112141 0.86 ESR2 (0.40) TDP2ESR2CYP3A4CYP2C9APP
SCHEMBL16280876 0.85 ESR2 (0.44) KDM1ACYP17A1ESR2CYP3A4CYP2C9
SCHEMBL2741559 0.85 ESR2 (0.44) KDM1ACYP17A1ESR2CYP3A4CYP2C9
SCHEMBL13112203 0.83 FASN (0.37) TDP2ESR2CYP3A4CYP2C9APP
SCHEMBL6455561 0.83 KDM1A (0.44) TDP2KDM1APTGS2NAAAPTGS1
SCHEMBL6455560 0.83 KDM1A (0.44) TDP2KDM1APTGS2NAAAPTGS1
SCHEMBL24661359 0.83 AKR1C3 (0.43) ESR2CYP3A4CYP2C9APP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110101270-A1 LIQUID-CRYSTALLINE MEDIUM MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2011-05-05 US disclosed